Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50029107
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281547((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 28nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281532((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 28nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281530((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 30nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281561((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 34nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281551((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 34nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281526((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 35nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281531((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 35nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281540((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 37nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281552((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 39nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281533((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 40nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281546((2S,3R)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50: 41nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281541((S)-6-Amino-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-amino-3-(...)
Affinity DataIC50: 41nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50080456(2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-p...)
Affinity DataIC50: 41nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281556((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 46nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281529((R)-1-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 57nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281528((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 59nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281537((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 60nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281550((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 65nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281535((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 65nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281545((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 75nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281557((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 77nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281534((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 78nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281560((2S,3S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50: 80nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281548((S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 98nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281553((S)-2-[(S)-2-((S)-2-{N-[2-(2-{N-[(S)-3-(4-Aminooxy...)
Affinity DataIC50: 107nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281558((R)-1-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 108nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281555((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 112nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281543((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 141nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281544(2-[2-(2-{2-[(S)-(S)-2-Amino-3-(4-hydroxy-phenyl)-1...)
Affinity DataIC50: 158nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281542((S)-3-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 167nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281539((2S,3S)-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hy...)
Affinity DataIC50: 168nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281559((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 189nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281554((S)-6-Amino-2-{(S)-2-[(S)-2-(2-{2-[(S)-2-amino-3-(...)
Affinity DataIC50: 201nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281536((S)-4-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 204nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281527((S)-3-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 214nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281538((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 223nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281549((S)-4-{(S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydrox...)
Affinity DataIC50: 315nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281525((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataIC50: 381nMAssay Description:Concentration required for 50% inhibition of [3H]DAGO binding to mu opioid receptor in crude rat brain homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article