Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029132
TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281663(3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-methyl-3,...)
Affinity DataKi:  0.210nMAssay Description:Tested in vitro for binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281663(3-Cyclopropylmethyl-6-ethyl-8-hydroxy-11-methyl-3,...)
Affinity DataKi:  1nMAssay Description:Tested in vitro for binding affinity against mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281660(N-Cyclohexyl-N-methyl-2-[2-(2-pyrrolidin-1-yl-etho...)
Affinity DataKi:  160nMAssay Description:Tested in vitro for binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281662(PD-146795 | 2-Benzofuran-4-yl-N-(tetrahydro-pyrrol...)
Affinity DataKi:  940nMAssay Description:Tested in vitro for binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281662(PD-146795 | 2-Benzofuran-4-yl-N-(tetrahydro-pyrrol...)
Affinity DataKi:  3.35E+3nMAssay Description:Tested in vitro for binding affinity against mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281660(N-Cyclohexyl-N-methyl-2-[2-(2-pyrrolidin-1-yl-etho...)
Affinity DataKi: >1.00E+4nMAssay Description:Tested in vitro for binding affinity against mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMu-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281661(PD-146884 | 2-Oxa-7,10-diaza-bicyclo[11.3.1]heptad...)
Affinity DataKi: >1.00E+4nMAssay Description:Tested in vitro for binding affinity against mu opioid receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetKappa-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50281661(PD-146884 | 2-Oxa-7,10-diaza-bicyclo[11.3.1]heptad...)
Affinity DataKi: >1.00E+4nMAssay Description:Tested in vitro for binding affinity against Opioid receptor kappa 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article