Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50029149
TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281791(Ac-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH | CHEMBL...)
Affinity DataKi:  0.0130nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataKi:  0.0180nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281781(Ac-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH | CHEMBL2645...)
Affinity DataKi:  0.0240nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281785((S)-2-{2-[(S)-2-{[(S)-1-((S)-2-{(S)-2-[((S)-1-Acet...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281793(Ac-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu...)
Affinity DataKi:  0.110nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281795(Ac-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH | CH...)
Affinity DataKi:  0.120nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50240844((S)-2-{2-[(S)-2-({(S)-1-[(S)-2-((S)-2-Acetylamino-...)
Affinity DataKi:  0.130nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50130880(pGlu-Leu-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-L...)
Affinity DataKi:  0.170nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281784(Ac-Tyr-Glu-Asn-Lys-Pro-Arg-Arg-Pro-Tyr-Ile-Leu-OH ...)
Affinity DataKi:  0.210nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281787((1S,4R)-2-{2-[2-({(S)-1-[(S)-2-((S)-2-Amino-propio...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281794((S)-2-{(2S,3R)-2-[(S)-2-{2-[2-((S)-2-(S)-Amino-5-g...)
Affinity DataKi:  0.920nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281782((1S,4R)-2-{2-[2-[((S)-{(S)-1-[2-((S)-2-Amino-5-gua...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281786(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281783((S)-1-[(S)-2-((S)-2-Amino-5-guanidino-pentanoylami...)
Affinity DataKi:  10nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281780((2S,5S)-2-{2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guan...)
Affinity DataKi:  110nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281790(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataKi:  200nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281789((S)-2-{2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataKi:  3.90E+3nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50281792((S)-1-[(S)-2-((S)-2-Amino-5-guanidino-pentanoylami...)
Affinity DataKi:  1.20E+4nMAssay Description:Inhibition of specific binding of [125I]-Tyr3-NT(1-13) to NT receptors in neonatal mouse whole brain (minus cerebellum)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article