Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50029175
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 0.150nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281984((S)-3-[(Z)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 0.300nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataIC50: 1.70nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281983((R)-3-[(Z)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 3.70nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]-Bolton Hunter CCK-26-33 to CCK-A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50212857(CHEMBL2115543)
Affinity DataIC50: 3.90nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]-Bolton Hunter CCK-26-33 to CCK-A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281984((S)-3-[(Z)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 13nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281984((S)-3-[(Z)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 18nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]-Bolton Hunter CCK-26-33 to CCK-A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50062005(PD-135666 | 3-[2-(2-Adamantan-2-yl-acetylamino)-3-...)
Affinity DataIC50: 30nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]-Bolton Hunter CCK-26-33 to CCK-A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50212857(CHEMBL2115543)
Affinity DataIC50: 60nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50281983((R)-3-[(Z)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 99nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]bolton Hunter CCK-26-33 to CCK-B receptor in the mouse cerebral cortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281984((S)-3-[(Z)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataIC50: 550nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]-Bolton Hunter CCK-26-33 to CCK-A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50449787(PD-134308 | CHEMBL2062154)
Affinity DataIC50: 4.30E+3nMAssay Description:Compound measured for half-maximal inhibition of specific binding of [125I]-Bolton Hunter CCK-26-33 to CCK-A receptor in the rat pancreas.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article