Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50029257
TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282741(2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282733(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282735(4'-(4-Oxo-2-propyl-8-thia-1,3-diaza-spiro[4.5]dec-...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282732(2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 2nMAssay Description:The compound was tested for the ability to displace 50% of totally specifically bound [125I]- Ang II from Angiotensin II receptor, type 1 siteMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282737(2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282740(5-Propyl-6-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282734(4'-(4,4-Dimethyl-5-oxo-2-propyl-4,5-dihydro-imidaz...)
Affinity DataIC50: 3nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282742(5,5-Dimethyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 4nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282730(2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 8nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282731(4'-(4-Oxo-2-propyl-1,3-diaza-spiro[4.4]non-1-en-3-...)
Affinity DataIC50: 9nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282738(2-Propyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylmet...)
Affinity DataIC50: 20nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282733(4'-(2-Butyl-4-oxo-1,3-diaza-spiro[4.4]non-1-en-3-y...)
Affinity DataIC50: 100nMAssay Description:The compound was tested for the ability to displace 50% of totally specifically bound [125I]- Ang II from Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282743(2-Methyl-5,5-diphenyl-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 100nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282735(4'-(4-Oxo-2-propyl-8-thia-1,3-diaza-spiro[4.5]dec-...)
Affinity DataIC50: 200nMAssay Description:The compound was tested for the ability to displace 50% of totally specifically bound [125I]- Ang II from Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282734(4'-(4,4-Dimethyl-5-oxo-2-propyl-4,5-dihydro-imidaz...)
Affinity DataIC50: 200nMAssay Description:The compound was tested for the ability to displace 50% of totally specifically bound [125I]- Ang II from Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282736(5,5-Diphenyl-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 300nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282731(4'-(4-Oxo-2-propyl-1,3-diaza-spiro[4.4]non-1-en-3-...)
Affinity DataIC50: 300nMAssay Description:The compound was tested for the ability to displace 50% of totally specifically bound [125I]- Ang II from Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282739(2,5,5-Triphenyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-...)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article