Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029269
TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282840((Z)-3-(3,5-Dibromo-4-hydroxy-phenyl)-2-pyridin-2-y...)
Affinity DataIC50: 1.05E+5nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282838((Z)-3-(3,5-Dibromo-4-hydroxy-phenyl)-2-pyridin-3-y...)
Affinity DataIC50: 1.68E+5nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282839((Z)-3-(3-Bromo-4-hydroxy-5-methoxy-phenyl)-2-pyrid...)
Affinity DataIC50: 2.42E+5nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50279881(CHEMBL300635 | CHEMBL69896 | 3-[(E)-2-(3,4,5-Trime...)
Affinity DataIC50: 5.16E+5nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50279879(2-[2-(3,4,5-Trimethoxy-phenyl)-vinyl]-pyridine | 2...)
Affinity DataIC50: 2.18E+6nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282837((Z)-3-(3,5-Dibromo-4-methoxy-phenyl)-2-pyridin-2-y...)
Affinity DataIC50: 2.53E+6nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282841(3-(3,5-Dibromo-4-hydroxy-phenyl)-2-pyridin-2-yl-pr...)
Affinity DataIC50: 2.09E+6nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetTyrosine-protein kinase Lck(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282842((Z)-3-(3,5-Dibromo-4-methoxy-phenyl)-2-pyridin-3-y...)
Affinity DataIC50: 2.53E+6nMAssay Description:Inhibition of p56 Lck tyrosine kinaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article