Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50029290
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016867((S)-6-Amino-2-((S)-2-{(R)-2-[(S)-2-amino-3-(4-hydr...)
Affinity DataKi:  0.380nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283041((R)-2-{2-[2-Amino-4-(2-{(S)-guanidino-1-(S)-2-[(R)...)
Affinity DataKi:  0.510nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283037([(S)-5-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283039([(S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283036([(S)-3-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283040([(S)-1-{(R)-1-[(S)-1-((S)-5-Amino-1-carbamoyl-pent...)
Affinity DataKi:  207nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283039([(S)-4-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  450nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283041((R)-2-{2-[2-Amino-4-(2-{(S)-guanidino-1-(S)-2-[(R)...)
Affinity DataKi:  497nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283035([(S)-3-Carbamoyl-3-((S)-2-{(S)-2-[(S)-2-trimethyla...)
Affinity DataKi:  1.30E+3nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283038([(S)-1-{(R)-1-[(S)-1-((S)-4-Amino-1-carbamoyl-buty...)
Affinity DataKi:  1.92E+3nMAssay Description:Binding affinity against mu-opioid receptor by using [3H]DAGO as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50016867((S)-6-Amino-2-((S)-2-{(R)-2-[(S)-2-amino-3-(4-hydr...)
Affinity DataKi:  2.36E+3nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283037([(S)-5-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  3.55E+3nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283036([(S)-3-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phe...)
Affinity DataKi:  5.86E+3nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283038([(S)-1-{(R)-1-[(S)-1-((S)-4-Amino-1-carbamoyl-buty...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283040([(S)-1-{(R)-1-[(S)-1-((S)-5-Amino-1-carbamoyl-pent...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283035([(S)-3-Carbamoyl-3-((S)-2-{(S)-2-[(S)-2-trimethyla...)
Affinity DataKi: >1.00E+5nMAssay Description:Binding affinity against delta-opioid receptor by using [3H]DADLE as radioligand in rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article