Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50029336
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataIC50: 8.5nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataIC50: 130nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50: 200nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50000092(Analog of 14-(Arylhydroxyamino)codeinone | 4-methy...)
Affinity DataIC50: 430nMAssay Description:Binding to delta opioid receptor by using [3H]DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283522(4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapentacycl...)
Affinity DataIC50: 530nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50: 640nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50: 910nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283521(10-(2-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50: 2.60E+3nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283519(4-methyl-10-(3-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50: 3.30E+3nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283523(4,10-dimethyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapent...)
Affinity DataIC50: 4.50E+3nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50: 5.10E+3nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283518(14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataIC50: 6.40E+3nMAssay Description:Binding to mu opioid receptor by using [3H]DAMGO as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283517(10-(3-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50: 7.40E+3nMAssay Description:Binding to delta opioid receptor by using [3H]DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50283516(1-[14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-...)
Affinity DataIC50: 7.90E+3nMAssay Description:Binding to delta opioid receptor by using [3H]DPDPE as radioligand in guinea pig brain minus cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283521(10-(2-furyl)-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4...)
Affinity DataIC50: 9.50E+3nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283522(4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapentacycl...)
Affinity DataIC50: 1.10E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283519(4-methyl-10-(3-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50: 1.50E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283525(4-methyl-10-(2-thienyl)-(1S,5R,13R,14S,17R)-12-oxa...)
Affinity DataIC50: 2.50E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283523(4,10-dimethyl-(1S,5R,13R,14S,17R)-12-oxa-4-azapent...)
Affinity DataIC50: 3.60E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283524(4-methyl-10-phenyl-(1S,5R,13R,14S,17R)-12-oxa-4-az...)
Affinity DataIC50: 7.60E+4nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283518(14-hydroxy-4-methyl-(1S,5R,13R,14S,17R)-12-oxa-4-a...)
Affinity DataIC50: 1.11E+5nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283520(10-benzo[b]thiophen-2-yl-4-methyl-(1S,5R,13R,14S,1...)
Affinity DataIC50: 1.26E+5nMAssay Description:Binding to kappa opioid receptor by using [3H]U-69593 as radioligand in guinea pig cerebellumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article