Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50029337
TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]-CGS- from Adenosine A2a receptor of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051232(8-(4-Fluoro-benzyl)-2-furan-2-yl-8H-pyrazolo[4,3-e...)
Affinity DataKi:  1.20nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051234(2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  1.40nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50007848(CHEMBL53737 | 8-Cyclopropyl-1,3-dipropyl-3,7-dihyd...)
Affinity DataKi:  1.5nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50094688(2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e]...)
Affinity DataKi:  1.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048466(CHEMBL17127 | SCH58261 | 2-(furan-2-yl)-7-phenethy...)
Affinity DataKi:  2.30nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051242(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]tria...)
Affinity DataKi:  2.40nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283532(2-(4-Fluoro-benzyl)-8-furan-2-yl-2H-[1,2,3]triazol...)
Affinity DataKi:  2.5nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051232(8-(4-Fluoro-benzyl)-2-furan-2-yl-8H-pyrazolo[4,3-e...)
Affinity DataKi:  3.30nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283529(3-Benzyl-8-furan-2-yl-3H-[1,2,3]triazolo[4,5-e][1,...)
Affinity DataKi:  4.60nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051234(2-(furan-2-yl)-8-phenethyl-8H-pyrazolo[4,3-e][1,2,...)
Affinity DataKi:  4.70nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283526(3-(3-Fluoro-benzyl)-8-furan-2-yl-3H-[1,2,3]triazol...)
Affinity DataKi:  4.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50094688(2-Furan-2-yl-8-(3-methyl-butyl)-8H-pyrazolo[4,3-e]...)
Affinity DataKi:  5.60nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283529(3-Benzyl-8-furan-2-yl-3H-[1,2,3]triazolo[4,5-e][1,...)
Affinity DataKi:  6.10nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50004566(CHEMBL268431 | 9-chloro-2-(furan-2-yl)-[1,2,4]tria...)
Affinity DataKi:  6.40nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283528(8-Furan-2-yl-3-phenethyl-3H-[1,2,3]triazolo[4,5-e]...)
Affinity DataKi:  6.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051227(7-Butyl-2-furan-2-yl-7H-pyrazolo[4,3-e][1,2,4]tria...)
Affinity DataKi:  8.90nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283527(3-(2-Fluoro-benzyl)-8-furan-2-yl-3H-[1,2,3]triazol...)
Affinity DataKi:  10.4nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283530(2-Furan-2-yl-7-(3-methyl-butyl)-7H-pyrazolo[4,3-e]...)
Affinity DataKi:  12nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283531(3-(4-Fluoro-benzyl)-8-furan-2-yl-3H-[1,2,3]triazol...)
Affinity DataKi:  13.7nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283527(3-(2-Fluoro-benzyl)-8-furan-2-yl-3H-[1,2,3]triazol...)
Affinity DataKi:  13.7nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283532(2-(4-Fluoro-benzyl)-8-furan-2-yl-2H-[1,2,3]triazol...)
Affinity DataKi:  18.3nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283526(3-(3-Fluoro-benzyl)-8-furan-2-yl-3H-[1,2,3]triazol...)
Affinity DataKi:  19nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051242(8-Butyl-2-furan-2-yl-8H-pyrazolo[4,3-e][1,2,4]tria...)
Affinity DataKi:  30.4nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283528(8-Furan-2-yl-3-phenethyl-3H-[1,2,3]triazolo[4,5-e]...)
Affinity DataKi:  42.4nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283531(3-(4-Fluoro-benzyl)-8-furan-2-yl-3H-[1,2,3]triazol...)
Affinity DataKi:  61.2nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051243(2-Furan-2-yl-7-methyl-7H-pyrazolo[4,3-e][1,2,4]tri...)
Affinity DataKi:  101nMAssay Description:Binding ability of adenosine A2a receptor by using [3H]-CGS- as radioligand in rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283530(2-Furan-2-yl-7-(3-methyl-butyl)-7H-pyrazolo[4,3-e]...)
Affinity DataKi:  116nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048466(CHEMBL17127 | SCH58261 | 2-(furan-2-yl)-7-phenethy...)
Affinity DataKi:  121nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051227(7-Butyl-2-furan-2-yl-7H-pyrazolo[4,3-e][1,2,4]tria...)
Affinity DataKi:  236nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A1(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051243(2-Furan-2-yl-7-methyl-7H-pyrazolo[4,3-e][1,2,4]tri...)
Affinity DataKi:  651nMAssay Description:Binding ability of adenosine A1 receptor by using [3H]CHA as radioligand in rat whole brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetAdenosine receptor A2a(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50007848(CHEMBL53737 | 8-Cyclopropyl-1,3-dipropyl-3,7-dihyd...)
Affinity DataKi:  706nMAssay Description:Displacement of [3H]-CGS- from Adenosine A2a receptor of rat striatal homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article