Compile Data Set for Download or QSAR
Report error Found 58 Enz. Inhib. hit(s) with all data for entry = 50029368
TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283831(N-tert-Butyl-2-[(3R,5S,7R)-7-(3-fluoro-phenyl)-2-o...)
Affinity DataIC50: 1nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283845(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283843(N-(2-Chloro-phenyl)-2-[(3R,5S,7R)-2-oxo-7-phenyl-5...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283832(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-p-toly...)
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283842(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-m-toly...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283838(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5-phenyl-7-m-toly...)
Affinity DataIC50: 1.60nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283826(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-fluoro-phenyl)-...)
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283827(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-methoxy-phenyl)...)
Affinity DataIC50: 2.20nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283839(N-tert-Butyl-2-[(3R,5S,7R)-7-(4-fluoro-phenyl)-2-o...)
Affinity DataIC50: 2.80nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283824(N-(1-Methyl-cyclohexyl)-2-[(3R,5S,7R)-2-oxo-7-phen...)
Affinity DataIC50: 4.40nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283825(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-o-toly...)
Affinity DataIC50: 7.80nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 8.10nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283841(N-(4-Chloro-phenyl)-2-[(3R,5S,7R)-2-oxo-7-phenyl-5...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283828(N-(3-Chloro-phenyl)-2-[(3R,5S,7R)-2-oxo-7-phenyl-5...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283840(N-tert-Butyl-2-[(3S,5S,7R)-2-oxo-5,7-diphenyl-3-(3...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283847(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-nitro-phenyl)-u...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283823(N-(1-tert-Butyl-2,2-dimethyl-propyl)-2-[(3R,5S,7R)...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283847(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-nitro-phenyl)-u...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283830(2-{(3R,5S,7R)-3-[3-(3-Ethyl-phenyl)-ureido]-2-oxo-...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283836(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283829(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-chloro-phenyl)-...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283833(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5,7-diphenyl-3-(3...)
Affinity DataIC50: 16nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283822(N-tert-Butyl-2-[(3R,5S,7R)-5-(2-ethyl-phenyl)-2-ox...)
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283843(N-(2-Chloro-phenyl)-2-[(3R,5S,7R)-2-oxo-7-phenyl-5...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283834(N-tert-Butyl-2-{(3R,5S,7R)-2-oxo-7-phenyl-5-o-toly...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283844(N-tert-Butyl-2-[(3R,5S,7R)-5-(2-methoxy-phenyl)-2-...)
Affinity DataIC50: 28nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283831(N-tert-Butyl-2-[(3R,5S,7R)-7-(3-fluoro-phenyl)-2-o...)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283826(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(3-fluoro-phenyl)-...)
Affinity DataIC50: 36nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283830(2-{(3R,5S,7R)-3-[3-(3-Ethyl-phenyl)-ureido]-2-oxo-...)
Affinity DataIC50: 38nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283836(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283837(N-tert-Butyl-2-[(3R,5S,7R)-5-(4-fluoro-phenyl)-2-o...)
Affinity DataIC50: 65nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283842(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-m-toly...)
Affinity DataIC50: 66nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283845(2-[(3R,5S,7R)-2-Oxo-7-phenyl-5-o-tolyl-3-(3-m-toly...)
Affinity DataIC50: 71nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283828(N-(3-Chloro-phenyl)-2-[(3R,5S,7R)-2-oxo-7-phenyl-5...)
Affinity DataIC50: 79nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283835(N-Isopropyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-o-tolyl...)
Affinity DataIC50: 80nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 86nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283827(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-methoxy-phenyl)...)
Affinity DataIC50: 87nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283829(N-tert-Butyl-2-{(3R,5S,7R)-3-[3-(4-chloro-phenyl)-...)
Affinity DataIC50: 117nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283824(N-(1-Methyl-cyclohexyl)-2-[(3R,5S,7R)-2-oxo-7-phen...)
Affinity DataIC50: 134nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283838(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5-phenyl-7-m-toly...)
Affinity DataIC50: 141nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283832(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-p-toly...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283839(N-tert-Butyl-2-[(3R,5S,7R)-7-(4-fluoro-phenyl)-2-o...)
Affinity DataIC50: 203nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283841(N-(4-Chloro-phenyl)-2-[(3R,5S,7R)-2-oxo-7-phenyl-5...)
Affinity DataIC50: 278nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283840(N-tert-Butyl-2-[(3S,5S,7R)-2-oxo-5,7-diphenyl-3-(3...)
Affinity DataIC50: 450nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283823(N-(1-tert-Butyl-2,2-dimethyl-propyl)-2-[(3R,5S,7R)...)
Affinity DataIC50: 453nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283825(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-o-toly...)
Affinity DataIC50: 527nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283825(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-o-toly...)
Affinity DataIC50: 527nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50283846(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-5-phenyl-7-p-toly...)
Affinity DataIC50: 560nMAssay Description:Inhibitory activity against cholecystokinin-B (CCK-B) receptor in cortex of male hartley guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283835(N-Isopropyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-o-tolyl...)
Affinity DataIC50: 560nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283825(N-tert-Butyl-2-[(3R,5S,7R)-2-oxo-7-phenyl-5-o-toly...)
Affinity DataIC50: 580nMAssay Description:Inhibitory activity against cholecystokinin-A (CCK-A) receptor in pancreas of guinea pig.More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

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