Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50029370
TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283867(N-Cyclohexylmethyl-N'-[3-(1H-imidazol-4-yl)-propyl...)
Affinity DataKi:  0.740nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283867(N-Cyclohexylmethyl-N'-[3-(1H-imidazol-4-yl)-propyl...)
Affinity DataKi:  0.794nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283869(N-[3-(1H-Imidazol-4-yl)-propyl]-N'-(4-iodo-benzyl)...)
Affinity DataKi:  1.58nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283869(N-[3-(1H-Imidazol-4-yl)-propyl]-N'-(4-iodo-benzyl)...)
Affinity DataKi:  1.60nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  3.98nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283874(N-Cyclohexyl-N'-[4-(1H-imidazol-4-yl)-butyl]-guani...)
Affinity DataKi:  5nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283874(N-Cyclohexyl-N'-[4-(1H-imidazol-4-yl)-butyl]-guani...)
Affinity DataKi:  5.01nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283871(N-(tert-Butoxy-carbonyl)-N'-cyclohexyl-N''-[4-(1H-...)
Affinity DataKi:  6.31nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283871(N-(tert-Butoxy-carbonyl)-N'-cyclohexyl-N''-[4-(1H-...)
Affinity DataKi:  7nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283868(N-(tert-Butoxy-carbonyl)-N'-cyclohexylmethyl-N''-[...)
Affinity DataKi:  9.5nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283868(N-(tert-Butoxy-carbonyl)-N'-cyclohexylmethyl-N''-[...)
Affinity DataKi:  10nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283873(N-Cyclohexylmethyl-N'-[3-(1H-imidazol-4-yl)-propyl...)
Affinity DataKi:  12.6nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283870(N-(tert-Butoxy-carbonyl)-N'-[3-(1H-imidazol-4-yl)-...)
Affinity DataKi:  12.6nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283870(N-(tert-Butoxy-carbonyl)-N'-[3-(1H-imidazol-4-yl)-...)
Affinity DataKi:  13nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283873(N-Cyclohexylmethyl-N'-[3-(1H-imidazol-4-yl)-propyl...)
Affinity DataKi:  13nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283876(N''-cyano-N-(cyclohexylmethyl)-N'-[3-(1H-imidazol-...)
Affinity DataKi:  19.9nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283876(N''-cyano-N-(cyclohexylmethyl)-N'-[3-(1H-imidazol-...)
Affinity DataKi:  22nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283875(N-Cyclohexylmethyl-N'-(ethoxy-hydroxy-methyl)-N''-...)
Affinity DataKi:  36nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283875(N-Cyclohexylmethyl-N'-(ethoxy-hydroxy-methyl)-N''-...)
Affinity DataKi:  39.8nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283872(N-[2-(1H-Imidazol-4-yl)-ethyl]-N'-phenethyl-guanid...)
Affinity DataKi:  100nMAssay Description:Antagonistic activity for Histamine H3 receptor on electrically evoked guinea-pig ileum contractionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetHistamine H3 receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50283872(N-[2-(1H-Imidazol-4-yl)-ethyl]-N'-phenethyl-guanid...)
Affinity DataKi:  110nMAssay Description:Antagonistic activity for Histamine H3 receptor binding in guinea pigMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article