Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 50029385
TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284007(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Ser-Val-Tyr-P...)
Affinity DataIC50: 60nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284006(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Aoa-Val-Tyr-Phe-C...)
Affinity DataIC50: 240nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284008(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Apa-Val-Tyr-Phe-C...)
Affinity DataIC50: 350nMAssay Description:Binding affinity against endothelin receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284011(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Asp-Lys-Glu-Val-T...)
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284007(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Ser-Val-Tyr-P...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284010(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Val-Tyr-Phe-C...)
Affinity DataIC50: 1.40E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284006(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Aoa-Val-Tyr-Phe-C...)
Affinity DataIC50: 1.60E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284014(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Val-Tyr-Phe-Cys) | CH...)
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284009(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Val-Tyr-Phe-Cys) ...)
Affinity DataIC50: 1.70E+3nMAssay Description:Binding affinity against Endothelin B receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284010(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Val-Tyr-Phe-C...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284006(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Aoa-Val-Tyr-Phe-C...)
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284008(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Apa-Val-Tyr-Phe-C...)
Affinity DataIC50: 1.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284010(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Val-Tyr-Phe-C...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284012(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Aha-Val-Tyr-Phe-C...)
Affinity DataIC50: 2.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284008(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Apa-Val-Tyr-Phe-C...)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284007(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Ser-Val-Tyr-P...)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284014(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Val-Tyr-Phe-Cys) | CH...)
Affinity DataIC50: 2.60E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284009(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Val-Tyr-Phe-Cys) ...)
Affinity DataIC50: 2.80E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284011(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Asp-Lys-Glu-Val-T...)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284009(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Val-Tyr-Phe-Cys) ...)
Affinity DataIC50: 3.80E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284014(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Val-Tyr-Phe-Cys) | CH...)
Affinity DataIC50: 6.50E+3nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284011(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Asp-Lys-Glu-Val-T...)
Affinity DataIC50: 7.10E+3nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284013(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Leu-Met-Asp-L...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against Endothelin A receptor in rabbit renal artery vascular smooth muscle membrane (ET-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284013(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Leu-Met-Asp-L...)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity against endothelin receptor in rat cerebellar membrane (ET-B) from adult blue laurie ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50284013(Trp-Ile-Ile-Asp-Leu-Hisc(Cys-Ser-Ser-Leu-Met-Asp-L...)
Affinity DataIC50: 4.90E+4nMAssay Description:In vitro binding affinity against Endothelin A receptor by using endothelin (ET-1) as radioligand in rat heart ventricleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article