Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50029402
TargetProlyl endopeptidase(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284127(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-2-carbonyl)-pyr...)
Affinity DataIC50: 3.10nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50037597(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-4-carbonyl)-pyr...)
Affinity DataIC50: 5.90nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284126((S)-1-[(S)-1-(4-Phenyl-butyryl)-pyrrolidine-2-carb...)
Affinity DataIC50: 8.70nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50088247(Oxo-{1-[1-(4-phenyl-butyryl)-pyrrolidine-2-carbony...)
Affinity DataIC50: 9.60nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50037599(4-Phenyl-1-{(S)-2-[(S)-2-(thiazole-5-carbonyl)-pyr...)
Affinity DataIC50: 646nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProlyl endopeptidase(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50037613(4-Phenyl-1-{(S)-2-[(S)-2-(thiophene-2-carbonyl)-py...)
Affinity DataIC50: 1.91E+3nMAssay Description:Compound was evaluated for the inhibition of Prolyl endopeptidase (PEP) from pig kidney using Z-Gly-Pro-p-nitroanilide as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article