Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50029405
TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284146([(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 14nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284148([(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 46nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284156([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 64nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284147([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 270nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50280054((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 350nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284160([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 430nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284161((E)-N-[(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine...)
Affinity DataIC50: 520nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284151(((2S,5S)-1-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-...)
Affinity DataIC50: 630nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284158(((2S,5S)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 840nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284152({(2S,5S)-5-Benzyl-1-[(S)-2-(2-1H-indol-3-yl-acetyl...)
Affinity DataIC50: 1.20E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284159(((2S,5S)-5-Benzyl-1-{(S)-2-[(1H-indole-3-carbonyl)...)
Affinity DataIC50: 1.40E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284144({(2S,5S)-5-Benzyl-1-[(S)-2-(2-1H-indol-3-yl-acetyl...)
Affinity DataIC50: 2.50E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284150(((2R,5S)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 2.80E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50280054((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 3.50E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284155(((2S,5R)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 3.60E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284157([(R)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 5.50E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284154(((2R,5R)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 6.30E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284152({(2S,5S)-5-Benzyl-1-[(S)-2-(2-1H-indol-3-yl-acetyl...)
Affinity DataIC50: 7.20E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284150(((2R,5S)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 7.40E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284151(((2S,5S)-1-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-...)
Affinity DataIC50: 8.20E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284153({(2S,5S)-5-Benzyl-1-[(S)-2-(3-1H-indol-3-yl-propio...)
Affinity DataIC50: 8.90E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284162(((2S,5S)-1-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-...)
Affinity DataIC50: 9.40E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284162(((2S,5S)-1-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-...)
Affinity DataIC50: 9.40E+3nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284149({[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-carbonyl)...)
Affinity DataIC50: 1.00E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284144({(2S,5S)-5-Benzyl-1-[(S)-2-(2-1H-indol-3-yl-acetyl...)
Affinity DataIC50: 1.30E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284146([(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 1.50E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284145(((2S,5S)-1-{(S)-2-[(S)-2-Amino-3-(1H-indol-3-yl)-p...)
Affinity DataIC50: 1.50E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284155(((2S,5R)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 1.70E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284156([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 1.80E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284149({[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-carbonyl)...)
Affinity DataIC50: 2.40E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284147([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 3.70E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284160([(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 3.80E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284148([(S)-1-[(S)-1-((R)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 3.90E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284145(((2S,5S)-1-{(S)-2-[(S)-2-Amino-3-(1H-indol-3-yl)-p...)
Affinity DataIC50: 5.10E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCholecystokinin receptor type A(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50284153({(2S,5S)-5-Benzyl-1-[(S)-2-(3-1H-indol-3-yl-propio...)
Affinity DataIC50: 5.60E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors on mouse pancreatic membranes (CCK-A)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284158(((2S,5S)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 6.10E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284154(((2R,5R)-5-Benzyl-1-{(S)-2-[(S)-2-tert-butoxycarbo...)
Affinity DataIC50: 7.00E+4nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284161((E)-N-[(S)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine...)
Affinity DataIC50: 1.00E+5nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284159(((2S,5S)-5-Benzyl-1-{(S)-2-[(1H-indole-3-carbonyl)...)
Affinity DataIC50: 1.00E+5nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284157([(R)-1-[(S)-1-((S)-3-Benzyl-5-oxo-piperazine-1-car...)
Affinity DataIC50: 1.00E+5nMAssay Description:Concentration producing half-maximal inhibition of specific binding of [125I]- CCK-8 to CCK receptors mouse forebrain membranes (CCK-B)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article