Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50029453
LigandPNGBDBM50012434(1-[3-(Quinolin-2-ylmethoxy)-phenyl]-hexan-1-ol | 1...)
Affinity DataIC50: 150nMAssay Description:Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemic cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50284680(3-Pyridin-3-ylmethyl-6-(quinolin-2-ylmethoxy)-chro...)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemic cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50070921(3-[6-(5-Fluoro-benzothiazol-2-ylmethoxy)-4-hydroxy...)
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of 5-Lipoxygenase (5-LO) in rat basophilic leukemic cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284680(3-Pyridin-3-ylmethyl-6-(quinolin-2-ylmethoxy)-chro...)
Affinity DataKi:  650nMAssay Description:Inhibition of [3H]LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284682(2-Benzyl-7-(quinolin-2-ylmethoxy)-1,2,3,4-tetrahyd...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibition of [3H]LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284681(2-Butyl-7-(quinolin-2-ylmethoxy)-1,2,3,4-tetrahydr...)
Affinity DataKi:  6.80E+3nMAssay Description:Inhibition of [3H]LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50012434(1-[3-(Quinolin-2-ylmethoxy)-phenyl]-hexan-1-ol | 1...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibition of [3H]LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50070921(3-[6-(5-Fluoro-benzothiazol-2-ylmethoxy)-4-hydroxy...)
Affinity DataKi:  2.40E+4nMAssay Description:Inhibition of [3H]LTD4 binding to LTD4 receptor in guinea pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article