Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50029456
TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284702(3-[(S)-2-[(S)-2-(3-tert-Butyl-ureido)-4-methyl-pen...)
Affinity DataIC50: 150nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membrane was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284693(3-{(S)-3-(1H-Indol-3-yl)-2-[(S)-4-methyl-2-(2-thio...)
Affinity DataIC50: 420nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membrane was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284692(3-[(S)-2-((S)-2-tert-Butoxycarbonylamino-4-methyl-...)
Affinity DataIC50: 420nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284695(3-[(S)-2-[(S)-2-(2-Cyclopentyl-acetylamino)-4-meth...)
Affinity DataIC50: 620nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membrane was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284700(3-{(S)-3-(1H-Indol-3-yl)-2-[(S)-4-methyl-2-(3-m-to...)
Affinity DataIC50: 2.10E+3nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284701(3-[(S)-2-{(S)-2-[3-(3-Chloro-phenyl)-ureido]-4-met...)
Affinity DataIC50: 2.10E+3nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284698(3-[(S)-2-[(S)-2-(3-Benzyl-ureido)-4-methyl-pentano...)
Affinity DataIC50: 3.20E+3nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284696(3-{(S)-3-(1H-Indol-3-yl)-2-[(S)-4-methyl-2-(3-meth...)
Affinity DataIC50: 3.90E+3nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membrane was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284694(3-[(S)-2-[(S)-2-(3,3-Dimethyl-butyrylamino)-4-meth...)
Affinity DataIC50: 6.70E+3nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284699(2-{3-(1H-Indol-3-yl)-2-[4-methyl-2-(3-methyl-butyr...)
Affinity DataIC50: 2.50E+4nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membrane was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetEndothelin-1 receptor(Pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284697(2-[2-[2-(2-Amino-3-methyl-butyrylamino)-4-methyl-p...)
Affinity DataIC50: 3.20E+4nMAssay Description:Binding affinity against ETA receptor in porcine aortic smooth muscle membrane was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article