Compile Data Set for Download or QSAR
Report error Found 38 Enz. Inhib. hit(s) with all data for entry = 50029476
TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284902((1-{(R)-1-{3-[(E)-2-(4-Cyclobutyl-thiazol-2-yl)-vi...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284902((1-{(R)-1-{3-[(E)-2-(4-Cyclobutyl-thiazol-2-yl)-vi...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284899({1-[(R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284899({1-[(R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284905((1-{(R)-1-{3-[(E)-2-(5,6-Difluoro-benzothiazol-2-y...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284895((1-{(R)-1-{3-[(E)-2-(4-Cyclopentyl-thiazol-2-yl)-v...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284895((1-{(R)-1-{3-[(E)-2-(4-Cyclopentyl-thiazol-2-yl)-v...)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284900([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284890((1-{(R)-1-{3-[(E)-2-(4-Cyclopropyl-thiazol-2-yl)-v...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284890((1-{(R)-1-{3-[(E)-2-(4-Cyclopropyl-thiazol-2-yl)-v...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284907([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284893((1-{(R)-1-{3-[(E)-2-(4-tert-Butyl-thiazol-2-yl)-vi...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284893((1-{(R)-1-{3-[(E)-2-(4-tert-Butyl-thiazol-2-yl)-vi...)
Affinity DataIC50: 2nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284896((1-{(R)-1-{3-[(E)-2-(4-Cyclohexyl-thiazol-2-yl)-vi...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284903((1-{(R)-1-{3-[(E)-2-(5,6-Dihydro-4H-cyclopentathia...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284903((1-{(R)-1-{3-[(E)-2-(5,6-Dihydro-4H-cyclopentathia...)
Affinity DataIC50: 3nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284901((1-{(R)-1-{3-[(E)-2-(5-Fluoro-benzothiazol-2-yl)-v...)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50013920(3-[(R)-{3-[(E)-2-(7-Chloro-quinolin-2-yl)-vinyl]-p...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284888((1-{(R)-1-(3-{(E)-2-[4-(4-Fluoro-phenyl)-thiazol-2...)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284888((1-{(R)-1-(3-{(E)-2-[4-(4-Fluoro-phenyl)-thiazol-2...)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284886([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284886([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284904((1-{(R)-1-{3-[(E)-2-(5-Chloro-benzothiazol-2-yl)-v...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284904((1-{(R)-1-{3-[(E)-2-(5-Chloro-benzothiazol-2-yl)-v...)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284887([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284887([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284897([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 12.8nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284897([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 13nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284908((1-{(R)-1-[3-((E)-2-Benzothiazol-2-yl-vinyl)-pheny...)
Affinity DataIC50: 17nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284906([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 42nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284898([1-((R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 48nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284891((1-{(R)-1-(3-{(E)-2-[4-(4-Chloro-phenyl)-thiazol-2...)
Affinity DataIC50: 79nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284891((1-{(R)-1-(3-{(E)-2-[4-(4-Chloro-phenyl)-thiazol-2...)
Affinity DataIC50: 79.3nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284889({1-[(R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 98.7nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284889({1-[(R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 99nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284892((1-{(R)-1-{3-[(E)-2-(5-Chloro-4-isopropyl-thiazol-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284892((1-{(R)-1-{3-[(E)-2-(5-Chloro-4-isopropyl-thiazol-...)
Affinity DataIC50: 170nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetCysteinyl leukotriene receptor 1(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50284894((1-{(R)-3-[2-(1-Hydroxy-1-methyl-ethyl)-phenyl]-1-...)
Affinity DataIC50: 381nMAssay Description:Inhibition of [3H]LTD4 binding on guinea-pig lung membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article