Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50029477
TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of human recombinant 92 kDa gelatinase MMP-9 at 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetInterstitial collagenase(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 2nMAssay Description:Inhibition of human recombinant interstitial collagenase MMP-1 at 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 28nMAssay Description:Inhibition of human recombinant matrix metalloprotease-3 (Stromelysin) at 100 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50284909((R)-3-Benzo[1,3]dioxol-5-yl-4-((S)-6-mercapto-5-me...)
Affinity DataIC50: 600nMAssay Description:Inhibition of human recombinant matrix metalloprotease-3 (Stromelysin) at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50213210(FUTOENONE)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of human recombinant matrix metalloprotease-3 (Stromelysin) at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article