Compile Data Set for Download or QSAR
Report error Found 51 Enz. Inhib. hit(s) with all data for entry = 50029524
TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50029600(CHEMBL42485 | 5-bromo-2-(4-fluorophenyl)-3-(4-(met...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285207(4-[2-(4-Fluoro-phenyl)-5-isopropyl-thiophen-3-yl]-...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285208(5-Bromo-3-(4-fluoro-phenyl)-2-(4-methanesulfonyl-p...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285228(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzenesulfo...)
Affinity DataIC50: 30nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285213(5-(4-Fluoro-phenyl)-4-(4-sulfamoyl-phenyl)-thiophe...)
Affinity DataIC50: 70nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285210(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzonitrile...)
Affinity DataIC50: 210nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285207(4-[2-(4-Fluoro-phenyl)-5-isopropyl-thiophen-3-yl]-...)
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285227(2-(4-Fluoro-phenyl)-3-(4-methanesulfonyl-phenyl)-t...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285223(2-(4-Fluoro-phenyl)-3-(4-methylsulfanyl-phenyl)-th...)
Affinity DataIC50: 340nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285216({4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-phenyl}-met...)
Affinity DataIC50: 350nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285220(4-[2-(4-Fluoro-phenyl)-5-(1-hydroxy-1-methyl-ethyl...)
Affinity DataIC50: 410nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285225(2-(4-Fluoro-phenyl)-3-(4-methaneselenonyl-phenyl)-...)
Affinity DataIC50: 550nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50029600(CHEMBL42485 | 5-bromo-2-(4-fluorophenyl)-3-(4-(met...)
Affinity DataIC50: 600nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285226(4-[3-(4-Fluoro-phenyl)-thiophen-2-yl]-benzenesulfo...)
Affinity DataIC50: 670nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285204(1-{4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-phenyl}-e...)
Affinity DataIC50: 750nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285215(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzaldehyde...)
Affinity DataIC50: 980nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285213(5-(4-Fluoro-phenyl)-4-(4-sulfamoyl-phenyl)-thiophe...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285208(5-Bromo-3-(4-fluoro-phenyl)-2-(4-methanesulfonyl-p...)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285228(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzenesulfo...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285211(4-[3-(4-Fluoro-phenyl)-5-(1-hydroxy-1-methyl-ethyl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285226(4-[3-(4-Fluoro-phenyl)-thiophen-2-yl]-benzenesulfo...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285217(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzamide | ...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285219(3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-t...)
Affinity DataIC50: 4.30E+3nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285220(4-[2-(4-Fluoro-phenyl)-5-(1-hydroxy-1-methyl-ethyl...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285206(N-Acetyl-4-[2-(4-fluoro-phenyl)-thiophen-3-yl]-ben...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285212(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-N-methyl-ben...)
Affinity DataIC50: 7.20E+3nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285209(2-(4-Fluoro-phenyl)-3-(4-methanesulfinyl-phenyl)-t...)
Affinity DataIC50: 1.50E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285221(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzoic acid...)
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285224(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzoic acid...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285222(4-{2-[4-(1-Hydroxy-1-methyl-ethyl)-phenyl]-thiophe...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285217(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzamide | ...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285205(3-(4-Ethanesulfonyl-phenyl)-2-(4-fluoro-phenyl)-th...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285210(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzonitrile...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285223(2-(4-Fluoro-phenyl)-3-(4-methylsulfanyl-phenyl)-th...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285209(2-(4-Fluoro-phenyl)-3-(4-methanesulfinyl-phenyl)-t...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285221(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzoic acid...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285204(1-{4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-phenyl}-e...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285218({4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-phenyl}-ace...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285216({4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-phenyl}-met...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285215(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzaldehyde...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 2(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285214(4-(4-Fluoro-phenyl)-5-(4-sulfamoyl-phenyl)-thiophe...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity against human COX-2 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285225(2-(4-Fluoro-phenyl)-3-(4-methaneselenonyl-phenyl)-...)
Affinity DataIC50: 3.20E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285219(3-(4-Fluoro-phenyl)-2-(4-methanesulfonyl-phenyl)-t...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285205(3-(4-Ethanesulfonyl-phenyl)-2-(4-fluoro-phenyl)-th...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285224(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-benzoic acid...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285211(4-[3-(4-Fluoro-phenyl)-5-(1-hydroxy-1-methyl-ethyl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285214(4-(4-Fluoro-phenyl)-5-(4-sulfamoyl-phenyl)-thiophe...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285222(4-{2-[4-(1-Hydroxy-1-methyl-ethyl)-phenyl]-thiophe...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285206(N-Acetyl-4-[2-(4-fluoro-phenyl)-thiophen-3-yl]-ben...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetProstaglandin G/H synthase 1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285212(4-[2-(4-Fluoro-phenyl)-thiophen-3-yl]-N-methyl-ben...)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibitory activity against human COX-1 expressed in baculovirus infected Sf9 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

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