Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50029536
LigandPNGBDBM50066068(N-Acenaphthen-5-yl-N'-(4-methoxy-naphthalen-1-yl)-...)
Affinity DataIC50: 1.31E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50285278(N,N'-Di-acenaphthen-5-yl-guanidine | CHEMBL307395)
Affinity DataIC50: 2.03E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM30705(SMR000058231 | CHEMBL744 | cid_5070 | MLS000069369...)
Affinity DataIC50: 2.20E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

LigandPNGBDBM50066430(CHEMBL28854 | 2-(4-Methyl-piperazin-1-yl)-5-(2,3,5...)
Affinity DataIC50: 2.55E+3nMAssay Description:Blockade of synaptosomal sodium channels, inhibition of [14C]guanidinium ion flux into CHO cells expressing Type II sodium channelMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article