Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50029543
TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285344([4-(7-Methyl-2-propyl-imidazo[4,5-b]pyridin-3-ylme...)
Affinity DataIC50: 5nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285349((2-Chloro-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50: 16nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285356((2-Ethoxy-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50: 18nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285345((4-Chloro-2-cyclohexyl-phenoxy)-(4-chloro-phenyl)-...)
Affinity DataIC50: 21nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285353((2,6-Dichloro-phenyl)-[4-(7-methyl-2-propyl-imidaz...)
Affinity DataIC50: 21nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285349((2-Chloro-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50: 22nMAssay Description:Tested in vitro for Angiotensin II receptor, type 2 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285346([4-(7-Methyl-2-propyl-imidazo[4,5-b]pyridin-3-ylme...)
Affinity DataIC50: 36nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285358((2-Methoxy-phenyl)-[4-(7-methyl-2-propyl-imidazo[4...)
Affinity DataIC50: 38nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50284459([4-(7-Methyl-2-propyl-imidazo[4,5-b]pyridin-3-ylme...)
Affinity DataIC50: 42nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285351([4-(7-Methyl-2-propyl-imidazo[4,5-b]pyridin-3-ylme...)
Affinity DataIC50: 57nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285355((3-Chloro-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50: 60nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285350(7-Methyl-3-{4-[phenyl-(1H-tetrazol-5-yl)-methoxy]-...)
Affinity DataIC50: 77nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285347((2-Hexyloxy-phenyl)-[4-(7-methyl-2-propyl-imidazo[...)
Affinity DataIC50: 80nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285357(2-{Carboxy-[4-(7-methyl-2-propyl-imidazo[4,5-b]pyr...)
Affinity DataIC50: 235nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285352(Cyclohexyl-[4-(7-methyl-2-propyl-imidazo[4,5-b]pyr...)
Affinity DataIC50: 325nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285354((4-Chloro-phenyl)-[4-(7-methyl-2-propyl-imidazo[4,...)
Affinity DataIC50: 530nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50285348(2-[4-(7-Methyl-2-propyl-imidazo[4,5-b]pyridin-3-yl...)
Affinity DataIC50: 840nMAssay Description:Tested in vitro for Angiotensin II receptor, type 1 binding affinity using rabbit aorta binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2010
Entry Details Article