Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50029860
Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051944(3-((1R,2S)-2-Dipropylamino-cyclopropyl)-phenol | C...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051956(2-((1R,2S)-2-Dipropylamino-cyclopropyl)-phenol | C...)
Affinity DataKi:  4.90nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50051950([(1S,2R)-2-(2-Methoxy-phenyl)-cyclopropyl]-dipropy...)
Affinity DataKi:  17nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288778(3-((1S,2R)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  58nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288773(3-((1S,2S)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  186nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288781([(1S,2S)-2-(2-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  239nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288780([(1S,2S)-2-(3-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  310nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288782(2-((1S,2R)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  379nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288775([(1R,2S)-2-(3-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  388nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288783(Diethyl-[(1S,2S)-2-(2-methoxy-phenyl)-cyclopropylm...)
Affinity DataKi:  431nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288776(2-((1S,2S)-2-Diethylaminomethyl-cyclopropyl)-pheno...)
Affinity DataKi:  506nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288774([(1R,2R)-2-(3-Methoxy-phenyl)-cyclopropyl]-dipropy...)
Affinity DataKi:  736nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288779(2-((1S,2S)-2-Dipropylaminomethyl-cyclopropyl)-phen...)
Affinity DataKi:  752nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288777([(1R,2S)-2-(2-Methoxy-phenyl)-cyclopropylmethyl]-d...)
Affinity DataKi:  998nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

Target5-hydroxytryptamine receptor 5A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50288772([(1R,2R)-2-(2-Methoxy-phenyl)-cyclopropyl]-dipropy...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of specific [3H]OH-DPAT binding at 5-hydroxytryptamine 1A receptor in rat hippocampal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article