Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50029998
LigandPNGBDBM50290085((2S,3R)-N*4*-((R)-2,2-Dimethyl-1-methylcarbamoyl-p...)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of human collagenase (MMP1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50290088((2S,3R)-N*1*-((R)-2,2-Dimethyl-1-methylcarbamoyl-p...)
Affinity DataIC50: 1nMAssay Description:Inhibition of human collagenase (MMP1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290089((2R,3R)-N*1*-[2,2-Dimethyl-1-((R)-methylcarbamoyl)...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human gelatinase B, MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50290089((2R,3R)-N*1*-[2,2-Dimethyl-1-((R)-methylcarbamoyl)...)
Affinity DataIC50: 2.60nMAssay Description:Inhibition of human collagenase (MMP1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290088((2S,3R)-N*1*-((R)-2,2-Dimethyl-1-methylcarbamoyl-p...)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of human gelatinase B, MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290085((2S,3R)-N*4*-((R)-2,2-Dimethyl-1-methylcarbamoyl-p...)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human gelatinase B, MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50290086(Ro-37-9790 | (R)-N*1*-[2,2-Dimethyl-1-((R)-methylc...)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human collagenase (MMP1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50290090((2S,3R)-3-Cyclopentylmethyl-N-hydroxy-4-oxo-4-pipe...)
Affinity DataIC50: 7nMAssay Description:Inhibition of human collagenase (MMP1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290085((2S,3R)-N*4*-((R)-2,2-Dimethyl-1-methylcarbamoyl-p...)
Affinity DataIC50: 9.10nMAssay Description:Inhibition of human stromelysin-1, MMP-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290086(Ro-37-9790 | (R)-N*1*-[2,2-Dimethyl-1-((R)-methylc...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human gelatinase B, MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

LigandPNGBDBM50290087((2S,3R)-5-Methyl-3-(piperidine-1-carbonyl)-2-(3,4,...)
Affinity DataIC50: 10nMAssay Description:Inhibition of human collagenase (MMP1)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290089((2R,3R)-N*1*-[2,2-Dimethyl-1-((R)-methylcarbamoyl)...)
Affinity DataIC50: 47nMAssay Description:Inhibition of human stromelysin-1, MMP-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290090((2S,3R)-3-Cyclopentylmethyl-N-hydroxy-4-oxo-4-pipe...)
Affinity DataIC50: 59nMAssay Description:Inhibition of human gelatinase B, MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290086(Ro-37-9790 | (R)-N*1*-[2,2-Dimethyl-1-((R)-methylc...)
Affinity DataIC50: 160nMAssay Description:Inhibition of human stromelysin-1, MMP-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetMatrix metalloproteinase-9(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290087((2S,3R)-5-Methyl-3-(piperidine-1-carbonyl)-2-(3,4,...)
Affinity DataIC50: 237nMAssay Description:Inhibition of human gelatinase B, MMP9More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290090((2S,3R)-3-Cyclopentylmethyl-N-hydroxy-4-oxo-4-pipe...)
Affinity DataIC50: 527nMAssay Description:Inhibition of human stromelysin-1, MMP-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetStromelysin-1(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290087((2S,3R)-5-Methyl-3-(piperidine-1-carbonyl)-2-(3,4,...)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of human stromelysin-1, MMP-3More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article