Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50030128
LigandPNGBDBM50006878(1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benzo[e]...)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50006842(CHEMBL37312 | 2-[2-(5-Bromo-1H-indol-3-yl)-ethyl]-...)
Affinity DataIC50: 9.30nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291402(3-{3-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-qu...)
Affinity DataIC50: 126nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50063620(1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 137nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291401(1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quina...)
Affinity DataIC50: 212nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291401(1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quina...)
Affinity DataIC50: 385nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50063624(1-(4-Bromo-phenyl)-3-{2-[3-(3-isopropoxy-phenyl)-4...)
Affinity DataIC50: 585nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291398(1-(4-Bromo-benzyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 652nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291399(1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quina...)
Affinity DataIC50: 674nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291399(1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quina...)
Affinity DataIC50: 691nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291404(1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quina...)
Affinity DataIC50: 879nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50063620(1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 984nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291403(1-((3,4-dihydro-3-(3-isopropoxyphenyl)-4-oxoquinaz...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50063660(1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50063660(1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291403(1-((3,4-dihydro-3-(3-isopropoxyphenyl)-4-oxoquinaz...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291402(3-{3-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-qu...)
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50063624(1-(4-Bromo-phenyl)-3-{2-[3-(3-isopropoxy-phenyl)-4...)
Affinity DataIC50: 1.63E+3nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291404(1-[3-(3-Isopropoxy-phenyl)-4-oxo-3,4-dihydro-quina...)
Affinity DataIC50: 1.64E+3nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291398(1-(4-Bromo-benzyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50291400(1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 6.93E+3nMAssay Description:Inhibition of specific binding of [125 I] Bolton Hunter CCK-8 to Cholecystokinin type A receptor in the rat pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50291400(1-(4-Bromo-phenyl)-3-[3-(3-isopropoxy-phenyl)-4-ox...)
Affinity DataIC50: 8.02E+3nMAssay Description:Inhibition of [125 I]CCK-8 binding to Cholecystokinin type B receptor of mouse cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article