Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 50034747
LigandPNGBDBM50000540(1-(3-Trifluoromethyl-phenyl)-4,5-dihydro-1H-pyrazo...)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50000540(1-(3-Trifluoromethyl-phenyl)-4,5-dihydro-1H-pyrazo...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281623(2-(4-fluorophenyl)-6-(2-naphthylsulfanyl)-1-hexana...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281622(2-(4-fluorophenyl)-6-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 4.10E+3nMAssay Description:Compound was tested for its ability to inhibit porcine pancreas phospholipase-A2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281621(6-[4-(tert-butyl)phenylsulfanyl]-2-(4-fluorophenyl...)
Affinity DataIC50: 4.80E+3nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281622(2-(4-fluorophenyl)-6-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 5.50E+3nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281625(2-(4-fluorophenyl)-7-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281622(2-(4-fluorophenyl)-6-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281626(2-(4-fluorophenyl)-5-(2-naphthylsulfanyl)-1-pentan...)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50281623(2-(4-fluorophenyl)-6-(2-naphthylsulfanyl)-1-hexana...)
Affinity DataIC50: 1.45E+4nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article
PDB3D3D Structure (crystal)
TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50281621(6-[4-(tert-butyl)phenylsulfanyl]-2-(4-fluorophenyl...)
Affinity DataIC50: 1.91E+4nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281626(2-(4-fluorophenyl)-5-(2-naphthylsulfanyl)-1-pentan...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50000540(1-(3-Trifluoromethyl-phenyl)-4,5-dihydro-1H-pyrazo...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281624(2-(4-fluorophenyl)-5-(4-methylphenylsulfanyl)-1-pe...)
Affinity DataIC50: 2.83E+4nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281624(2-(4-fluorophenyl)-5-(4-methylphenylsulfanyl)-1-pe...)
Affinity DataIC50: 2.83E+4nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281625(2-(4-fluorophenyl)-7-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281624(2-(4-fluorophenyl)-5-(4-methylphenylsulfanyl)-1-pe...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281624(2-(4-fluorophenyl)-5-(4-methylphenylsulfanyl)-1-pe...)
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50281626(2-(4-fluorophenyl)-5-(2-naphthylsulfanyl)-1-pentan...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50281625(2-(4-fluorophenyl)-7-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 4.80E+4nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50281622(2-(4-fluorophenyl)-6-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 4.87E+4nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50015214(N-(4-Hydroxy-phenyl)-acetamide | 6-chloro-2-methox...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50015214(N-(4-Hydroxy-phenyl)-acetamide | 6-chloro-2-methox...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281623(2-(4-fluorophenyl)-6-(2-naphthylsulfanyl)-1-hexana...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50015214(N-(4-Hydroxy-phenyl)-acetamide | 6-chloro-2-methox...)
Affinity DataIC50: 1.30E+5nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50281624(2-(4-fluorophenyl)-5-(4-methylphenylsulfanyl)-1-pe...)
Affinity DataIC50: 1.97E+5nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin G/H synthase 1/2(Sheep)
TBA

Curated by ChEMBL
LigandPNGBDBM50281624(2-(4-fluorophenyl)-5-(4-methylphenylsulfanyl)-1-pe...)
Affinity DataIC50: 2.15E+5nMAssay Description:Inhibition of ovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281621(6-[4-(tert-butyl)phenylsulfanyl]-2-(4-fluorophenyl...)
Affinity DataIC50: 2.30E+5nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibition of rat basophilic leukemia cell 5-lipoxygenaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM17638(indometacin | Indocin | 2-{1-[(4-chlorophenyl)carb...)
Affinity DataIC50: 2.50E+5nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetProstaglandin-H2 D-isomerase(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50281622(2-(4-fluorophenyl)-6-(4-methylphenylsulfanyl)-1-he...)
Affinity DataIC50: 2.80E+5nMAssay Description:Compound was tested for its ability to inhibit bovine seminal vesicle prostaglandin synthetaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetPhospholipase A2(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM18207(dexamethasone (tetramethyl-rhodamine conjugated ) ...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibitory activity against polymorphonuclear cell phospholipase-A2 in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article