Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50034749
TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281699(5-Dipentylcarbamoyl-5-[((R)-naphthalene-2-carbonyl...)
Affinity DataIC50: 30nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50005459(CHEMBL9485 | CR 1409 | 4-(3,4-Dichloro-benzoylamin...)
Affinity DataIC50: 50nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281696(N-[1-(3-Aza-spiro[5.5]undecane-3-carbonyl)-4-(4-me...)
Affinity DataIC50: 600nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281693(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-4-(4-meth...)
Affinity DataIC50: 700nMAssay Description:The compound was tested for its activity to inhibit the specific binding of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50048772((R)-5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-b...)
Affinity DataIC50: 1.40E+3nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281690(Naphthalene-2-carboxylic acid [1-dipentylcarbamoyl...)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281697(3,4-Dichloro-N-[1-dipentylcarbamoyl-4-(4-methyl-pi...)
Affinity DataIC50: 1.80E+3nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281694(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-diet...)
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281692(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-morp...)
Affinity DataIC50: 2.80E+3nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281695(N-{1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-[(E)-2-...)
Affinity DataIC50: 3.30E+3nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281699(5-Dipentylcarbamoyl-5-[((R)-naphthalene-2-carbonyl...)
Affinity DataIC50: 3.80E+3nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281696(N-[1-(3-Aza-spiro[5.5]undecane-3-carbonyl)-4-(4-me...)
Affinity DataIC50: 5.00E+3nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50005459(CHEMBL9485 | CR 1409 | 4-(3,4-Dichloro-benzoylamin...)
Affinity DataIC50: 5.60E+3nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281693(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-4-(4-meth...)
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281693(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-4-(4-meth...)
Affinity DataIC50: 6.60E+3nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281698(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-dime...)
Affinity DataIC50: 1.25E+4nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281695(N-{1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-[(E)-2-...)
Affinity DataIC50: 1.28E+4nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50048772((R)-5-(8-Aza-spiro[4.5]dec-8-yl)-4-(3,5-dichloro-b...)
Affinity DataIC50: 1.35E+4nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281692(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-morp...)
Affinity DataIC50: 1.39E+4nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281690(Naphthalene-2-carboxylic acid [1-dipentylcarbamoyl...)
Affinity DataIC50: 1.60E+4nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281694(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-diet...)
Affinity DataIC50: 1.85E+4nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281698(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-3-(2-dime...)
Affinity DataIC50: 3.13E+4nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281700(2-(3-Chloro-benzoylamino)-pentanedioic acid 1-[(2-...)
Affinity DataIC50: 4.22E+4nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50281691(3-Chloro-N-[1-(3,3-dimethyl-butylcarbamoyl)-4-(4-m...)
Affinity DataIC50: 4.88E+4nMAssay Description:Displacement of [125I](BH)-CCK-8 to Cholecystokinin type A receptor in rat pancreatic aciniMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281697(3,4-Dichloro-N-[1-dipentylcarbamoyl-4-(4-methyl-pi...)
Affinity DataIC50: 5.00E+4nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281691(3-Chloro-N-[1-(3,3-dimethyl-butylcarbamoyl)-4-(4-m...)
Affinity DataIC50: 1.04E+5nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50281693(N-[1-(8-Aza-spiro[4.5]decane-8-carbonyl)-4-(4-meth...)
Affinity DataIC50: 1.21E+5nMAssay Description:Displacement of [3H](N-methyl-N-leucine)-CCK-8 to Cholecystokinin type B receptor of guinea pig brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article