Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50034767
TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50403247(CHEMBL2079791)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282613(6-{2-Cyclopropyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50403246(CHEMBL2079787)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50403245(CHEMBL2079788)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50403242(CHEMBL2079790)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM82258(NSC_3961 | CAS_114798-26-4 | Losartan)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50403243(CHEMBL2079789)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282616(6-{2-Cyclopropyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50403244(CHEMBL2079785)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282611((3-{2-Cyclopropyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50: 4nMAssay Description:Inhibitory activity against Angiotensin II receptor, type 1 induced contractions in isolated rabbit aortic ringsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50282626(6-{2-Butyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 22nMAssay Description:Concentration required for 50% inhibition of binding against Angiotensin II receptor, type 1 in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50282629(6-{2-Butyl-1-[2'-(1H-tetrazol-5-yl)-biphenyl-4-ylm...)
Affinity DataIC50: 161nMAssay Description:Concentration required for 50% inhibition of binding against Angiotensin II receptor, type 1 in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50282623(6-{2-(4-Methoxy-phenyl)-1-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataIC50: 5.50E+3nMAssay Description:Concentration required for 50% inhibition of binding against Angiotensin II receptor, type 1 in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50282621(6-(2-Butyl-1H-benzoimidazol-5-yl)-5-methyl-2-[2'-(...)
Affinity DataIC50: 7.00E+3nMAssay Description:Concentration required for 50% inhibition of binding against Angiotensin II receptor, type 1 in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50282617(6-[2-(4-methoxyphenyl)-1H-benzimidazol-5-yl]-5-met...)
Affinity DataIC50: 1.70E+4nMAssay Description:Concentration required for 50% inhibition of binding against Angiotensin II receptor, type 1 in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50282615(6-[2-(4-Methoxy-phenyl)-1H-benzoimidazol-5-yl]-5-m...)
Affinity DataIC50: 5.40E+4nMAssay Description:Concentration required for 50% inhibition of binding against Angiotensin II receptor, type 1 in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50282612(6-(2-Butyl-1H-benzoimidazol-5-yl)-5-methyl-4,5-dih...)
Affinity DataIC50: 1.00E+6nMAssay Description:Concentration required for 50% inhibition of binding against Angiotensin II receptor, type 1 in bovine adrenal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article