Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50034768
TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282708(Thiophene-2-carboxylic acid benzyl-{2-ethyl-4-oxo-...)
Affinity DataIC50: 0.0600nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50041969(3-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 0.100nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282710(N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)...)
Affinity DataIC50: 0.220nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282702(Thiophene-2-carboxylic acid benzyl-{2-isopropyl-4-...)
Affinity DataIC50: 0.240nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282705(N-Benzyl-N-{2-isopropyl-4-oxo-3-[2'-(1H-tetrazol-5...)
Affinity DataIC50: 0.350nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282704(N-(2-Chloro-benzyl)-N-{2-ethyl-4-oxo-3-[2'-(1H-tet...)
Affinity DataIC50: 0.460nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50049182(PD-126055 | (S)-5-Benzyloxy-2-diphenylacetyl-6-met...)
Affinity DataIC50: 0.580nMAssay Description:In vitro binding affinity of compound was measured against angiotensin II (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article
PDB3D3D Structure (crystal)
TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50041967(Benzyl-{4-oxo-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bi...)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282699(N-{4-Oxo-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50: 0.700nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282700(N-(2-Chloro-benzyl)-N-{2-methyl-4-oxo-3-[2'-(1H-te...)
Affinity DataIC50: 0.740nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282706(N-{2-Ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282703(N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282701(N-Benzyl-N-{2-methyl-4-oxo-3-[2'-(1H-tetrazol-5-yl...)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50280907(L-159686 | (S)-1,4-Bis-diphenylcarbamoyl-piperazin...)
Affinity DataIC50: 1.5nMAssay Description:In vitro binding affinity of compound was measured against Angiotensin II receptor, type 2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282699(N-{4-Oxo-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bipheny...)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282707(Benzyl-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 3.30nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50041967(Benzyl-{4-oxo-2-propyl-3-[2'-(1H-tetrazol-5-yl)-bi...)
Affinity DataIC50: 4.90nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282709(Benzyl-{2-butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 5.10nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50282396(PD-123319 | (S)-1-(4-Dimethylamino-3-methyl-benzyl...)
Affinity DataIC50: 6.90nMAssay Description:In vitro binding affinity of compound was measured against angiotensin II (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50049192((S)-2-Diphenylacetyl-6-phenyl-1,2,3,4-tetrahydro-i...)
Affinity DataIC50: 30nMAssay Description:In vitro binding affinity of compound was measured against angiotensin II (AT2) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282709(Benzyl-{2-butyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 33nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282702(Thiophene-2-carboxylic acid benzyl-{2-isopropyl-4-...)
Affinity DataIC50: 42nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282710(N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)...)
Affinity DataIC50: 72nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282706(N-{2-Ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 79nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282707(Benzyl-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)-bip...)
Affinity DataIC50: 160nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282703(N-Benzyl-N-{2-ethyl-4-oxo-3-[2'-(1H-tetrazol-5-yl)...)
Affinity DataIC50: 170nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282708(Thiophene-2-carboxylic acid benzyl-{2-ethyl-4-oxo-...)
Affinity DataIC50: 200nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282704(N-(2-Chloro-benzyl)-N-{2-ethyl-4-oxo-3-[2'-(1H-tet...)
Affinity DataIC50: 410nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282701(N-Benzyl-N-{2-methyl-4-oxo-3-[2'-(1H-tetrazol-5-yl...)
Affinity DataIC50: 590nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282700(N-(2-Chloro-benzyl)-N-{2-methyl-4-oxo-3-[2'-(1H-te...)
Affinity DataIC50: 820nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-1 angiotensin II receptor(Rabbit)
TBA

Curated by ChEMBL
LigandPNGBDBM50282705(N-Benzyl-N-{2-isopropyl-4-oxo-3-[2'-(1H-tetrazol-5...)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from type 1 Angiotensin II receptor of rabbit aorta membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetType-2 angiotensin II receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50041969(3-{2-Butyl-4-oxo-3-[2'-(2H-tetrazol-5-yl)-biphenyl...)
Affinity DataIC50: 4.50E+3nMAssay Description:Displacement of [125 I]Sar1Ile8-AII from AT2 receptor of rat midbrain membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article