Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50034802
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50326659(3,10-dimethoxy-17-methyl-(10S)-17-azatetracyclo[7....)
Affinity DataKi:  0.700nMAssay Description:Binding affinity by its ability to displace [3H]DAMGO from mu receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50285003(3,10-dimethoxy-17-phenethyl-17-azatetracyclo[7.5.3...)
Affinity DataKi:  0.900nMAssay Description:Binding affinity by its ability to displace [3H]DAMGO from mu receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50326659(3,10-dimethoxy-17-methyl-(10S)-17-azatetracyclo[7....)
Affinity DataKi:  1.5nMAssay Description:Binding affinity by its ability to displace [3H]-U-69,593 from kappa receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50148071(Naltrindole analogue | 17-cyclopropylmethyl-3,10-d...)
Affinity DataKi:  24nMAssay Description:Binding affinity by its ability to displace [3H]DAMGO from mu receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50326659(3,10-dimethoxy-17-methyl-(10S)-17-azatetracyclo[7....)
Affinity DataKi:  46nMAssay Description:Binding affinity by its ability to displace [3H]DPDPE from delta receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50285003(3,10-dimethoxy-17-phenethyl-17-azatetracyclo[7.5.3...)
Affinity DataKi:  49nMAssay Description:Binding affinity by its ability to displace [3H]DPDPE from delta receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50148071(Naltrindole analogue | 17-cyclopropylmethyl-3,10-d...)
Affinity DataKi:  61nMAssay Description:Binding affinity by its ability to displace [3H]-U-69,593 from kappa receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetDelta-type opioid receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50148071(Naltrindole analogue | 17-cyclopropylmethyl-3,10-d...)
Affinity DataKi:  105nMAssay Description:Binding affinity by its ability to displace [3H]DPDPE from delta receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article

TargetKappa-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50285003(3,10-dimethoxy-17-phenethyl-17-azatetracyclo[7.5.3...)
Affinity DataKi:  690nMAssay Description:Binding affinity by its ability to displace [3H]-U-69,593 from kappa receptor in homogenates of guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2012
Entry Details Article