Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50034811
LigandPNGBDBM50285623((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKd:  0.25nMAssay Description:The equilibrium binding constant to guinea pig cerebral cortex membranes was measuredMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

LigandPNGBDBM50285625(PD-142251 | (R)-3-[2-((R)-Adamantan-2-yloxycarbony...)
Affinity DataKd:  8.10nMAssay Description:The equilibrium binding constant to pig cerebral cortex membranes was measuredMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

LigandPNGBDBM50285624((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKd:  0.110nMAssay Description:The equilibrium binding constant to guinea pig cerebral cortex membranes was measuredMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

LigandPNGBDBM50285623((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of binding of [125I]-PD 142308 to CCK-B receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

LigandPNGBDBM50285623((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  0.520nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex membrane using [125I]bolton assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

LigandPNGBDBM50285625(PD-142251 | (R)-3-[2-((R)-Adamantan-2-yloxycarbony...)
Affinity DataKi:  0.880nMAssay Description:Binding affinity towards CCK-B receptor in mouse cerebral cortex membrane using [125I]bolton assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataKi:  15nMAssay Description:Inhibition of binding of [125I]-PD 142308 to CCK-B receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataKi:  52nMAssay Description:Inhibition of binding of [125I]-PD 142251 to CCK-B receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50285623((R)-3-[(R)-2-(Adamantan-2-yloxycarbonylamino)-3-(1...)
Affinity DataKi:  158nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas membrane using Hunter labelled CCK-8S assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetCholecystokinin receptor type A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50285625(PD-142251 | (R)-3-[2-((R)-Adamantan-2-yloxycarbony...)
Affinity DataKi:  392nMAssay Description:Binding affinity towards CCK-A receptor in rat pancreas membrane using Hunter labelled CCK-8S assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article