Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50034816
TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataKi:  18nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286239([(1S,4R,5R)-11-((S)-Isobutyl)-14-((R)-isopropyl)-8...)
Affinity DataKi:  224nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286244([(1S,4R,5R)-8-Benzyl-11-((S)-isobutyl)-14-((R)-iso...)
Affinity DataKi:  2.40E+3nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286238({8-[(1H-Indole-2-carbonyl)-amino]-11-oxo-5-propyl-...)
Affinity DataKi:  6.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286234([8-(2-1H-Indol-3-yl-acetylamino)-11-oxo-5-propyl-5...)
Affinity DataKi:  7.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50329850((R)-3-Amino-4-[(S)-2-((R)-1-{(S)-1-[(R)-1-(1H-indo...)
Affinity DataKi:  7.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286237([8-(Naphthalen-1-ylmethoxy)-11-oxo-5-propyl-5,11-d...)
Affinity DataKi:  7.00E+3nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286243([8-(Naphthalen-1-ylmethoxy)-11-oxo-5,11-dihydro-di...)
Affinity DataKi:  8.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286240({8-[(Naphthalen-1-ylmethyl)-amino]-11-oxo-5-propyl...)
Affinity DataKi:  9.00E+3nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286242({8-[(1H-Indole-3-carbonyl)-amino]-11-oxo-5-propyl-...)
Affinity DataKi:  1.10E+4nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286235([8-(1H-Indol-3-ylmethyl)-11-oxo-5-propyl-5,11-dihy...)
Affinity DataKi:  1.20E+4nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286234([8-(2-1H-Indol-3-yl-acetylamino)-11-oxo-5-propyl-5...)
Affinity DataKi:  1.40E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286240({8-[(Naphthalen-1-ylmethyl)-amino]-11-oxo-5-propyl...)
Affinity DataKi:  1.70E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286243([8-(Naphthalen-1-ylmethoxy)-11-oxo-5,11-dihydro-di...)
Affinity DataKi:  2.80E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286238({8-[(1H-Indole-2-carbonyl)-amino]-11-oxo-5-propyl-...)
Affinity DataKi:  3.30E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286235([8-(1H-Indol-3-ylmethyl)-11-oxo-5-propyl-5,11-dihy...)
Affinity DataKi:  4.10E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286237([8-(Naphthalen-1-ylmethoxy)-11-oxo-5-propyl-5,11-d...)
Affinity DataKi:  6.00E+4nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286242({8-[(1H-Indole-3-carbonyl)-amino]-11-oxo-5-propyl-...)
Affinity DataKi:  8.00E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286236({8-[(Naphthalene-1-carbonyl)-amino]-11-oxo-5-propy...)
Affinity DataKi:  8.30E+4nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin receptor type B(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50286241((8-Benzyloxy-11-oxo-5,11-dihydro-dibenzo[b,e][1,4]...)
Affinity DataKi: >1.00E+5nMAssay Description:Affinity against ET B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetEndothelin-1 receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50286241((8-Benzyloxy-11-oxo-5,11-dihydro-dibenzo[b,e][1,4]...)
Affinity DataKi:  1.09E+5nMAssay Description:Affinity against ET A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article