Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50034831
TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286859(2-{2-[(S)-2-({1-[(S)-6-Amino-2-((S)-(S)-2,6-diamin...)
Affinity DataKi:  0.0600nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50240339(CHEMBL266571 | Neurotensin 2 | 2-{(R)-(S)-2-[(S)-2...)
Affinity DataKi:  0.0640nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286864((S)-2-{(S)-2-[(S)-2-({(R)-1-[5-Guanidino-2-(3-guan...)
Affinity DataKi:  0.100nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50366427(CHEMBL1793865)
Affinity DataKi:  0.150nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286868((1S,2S,4S)-2-{2-[(S)-2-({1-[6-Amino-2-(2,6-diamino...)
Affinity DataKi:  0.400nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50240845(2-{(S)-2-[2-({(S)-1-[(S)-2-((S)-2-Amino-5-guanidin...)
Affinity DataKi:  0.520nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286866(2-{2-[(S)-2-({1-[(S)-6-Amino-2-((S)-2,6-diamino-he...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286861((S)-2-{(S)-2-[(S)-2-({(R)-1-[6-Amino-2-(4-amino-bu...)
Affinity DataKi:  3.80nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286863((S)-2-{(S)-2-[(S)-2-({(R)-1-[5-Amino-2-(3-amino-pr...)
Affinity DataKi:  17nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286865((S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataKi:  17nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286867((S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-(6-amin...)
Affinity DataKi:  27nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286869((S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-((S)-2,...)
Affinity DataKi:  31nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286858((S)-2-{(S)-2-[(S)-2-{[(S)-1-((S)-2,6-Diamino-hexan...)
Affinity DataKi:  60nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeurotensin receptor type 1(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50286862((S)-2-{(S)-2-[(S)-2-({(R)-1-[(S)-6-Amino-2-((S)-2-...)
Affinity DataKi:  437nMAssay Description:Compound was tested in vitro for its binding affinity against Neurotensin Receptor after peripheral administrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article