Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50042149
Target5-hydroxytryptamine receptor 1A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataIC50: 0.300nMAssay Description:In Vitro Binding affinity againist 5-HT1A receptor by displacing [3H]8-OH-DPAT from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 1D(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataIC50: 3.40nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 1D receptor by displacing [125I]GTI from pig caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421346(CHEMBL19114)
Affinity DataIC50: 4.60nMAssay Description:In Vitro Binding affinity againist 5-HT1A receptor by displacing [3H]8-OH-DPAT from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421348(CHEMBL18710)
Affinity DataIC50: 9.10nMAssay Description:In Vitro Binding affinity againist 5-HT1A receptor by displacing [3H]8-OH-DPAT from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 1D(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421346(CHEMBL19114)
Affinity DataIC50: 43nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 1D receptor by displacing [125I]GTI from pig caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 1A(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421347(CHEMBL18928)
Affinity DataIC50: 72nMAssay Description:In Vitro Binding affinity againist 5-HT1A receptor by displacing [3H]8-OH-DPAT from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 1D(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421348(CHEMBL18710)
Affinity DataIC50: 151nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 1D receptor by displacing [125I]GTI from pig caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 2C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataIC50: 589nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 2C receptor by displacing [3H]mesulergine from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 2C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421346(CHEMBL19114)
Affinity DataIC50: 661nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 2C receptor by displacing [3H]mesulergine from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 1D(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421347(CHEMBL18928)
Affinity DataIC50: 776nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 1D receptor by displacing [125I]GTI from pig caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 2A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50421346(CHEMBL19114)
Affinity DataIC50: 1.70E+3nMAssay Description:In Vitro Binding affinity againist 5-HT2A receptor by displacing [3H]-DOB from rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 2A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50421348(CHEMBL18710)
Affinity DataIC50: 3.39E+3nMAssay Description:In Vitro Binding affinity againist 5-HT2A receptor by displacing [3H]-DOB from rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 3A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50421348(CHEMBL18710)
Affinity DataIC50: 3.98E+3nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 3 receptor by displacing [3H]-Q-ICS 205-930 from rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 2C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421348(CHEMBL18710)
Affinity DataIC50: 4.17E+3nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 2C receptor by displacing [3H]mesulergine from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 3A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50421347(CHEMBL18928)
Affinity DataIC50: 4.27E+3nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 3 receptor by displacing [3H]-Q-ICS 205-930 from rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 3A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50421346(CHEMBL19114)
Affinity DataIC50: 7.41E+3nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 3 receptor by displacing [3H]-Q-ICS 205-930 from rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 2C(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50421347(CHEMBL18928)
Affinity DataIC50: 8.13E+3nMAssay Description:In Vitro Binding affinity againist 5-hydroxytryptamine 2C receptor by displacing [3H]mesulergine from pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article

Target5-hydroxytryptamine receptor 2A(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM21392([3H]-5-carboxamidotryptamine | CHEMBL18840 | 5-car...)
Affinity DataIC50: 2.19E+4nMAssay Description:In Vitro Binding affinity againist 5-HT2A receptor by displacing [3H]-DOB from rat cortex homogenatesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/22/2013
Entry Details Article