Compile Data Set for Download or QSAR
Report error Found 76 Enz. Inhib. hit(s) with all data for entry = 50035521
LigandPNGBDBM50366495(CHEMBL1255588 | (+)butaclamol)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM21397(8-[4-(4-fluorophenyl)-4-oxidanylidene-butyl]-1-phe...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50017721(5-(1-methylpiperidylidene-4)-5H-dibenzo(a,d)cyclop...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026964(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-11H-benz...)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026964(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-11H-benz...)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026974(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-6,11-dih...)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026974(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-6,11-dih...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026970(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-6,11-di...)
Affinity DataKi:  8.20nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026964(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-11H-benz...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026970(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-6,11-di...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026974(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-6,11-dih...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026971(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026973(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026972(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026967(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026963(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026972(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026963(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026967(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026973(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026964(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-11H-benz...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026964(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-11H-benz...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026970(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-6,11-di...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026968(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-11H-ben...)
Affinity DataKi:  20nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026971(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  21nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026967(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026969(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]LSD radioligand binding at the serotonin-1 binding site of rat cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026971(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026972(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026971(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026963(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026971(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026973(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  36nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026974(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-6,11-dih...)
Affinity DataKi:  44nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026970(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-6,11-di...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026969(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026974(9-Bromo-11-(1-methyl-piperidin-4-ylidene)-6,11-dih...)
Affinity DataKi:  60nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50017721(5-(1-methylpiperidylidene-4)-5H-dibenzo(a,d)cyclop...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026970(9-Chloro-11-(1-methyl-piperidin-4-ylidene)-6,11-di...)
Affinity DataKi:  80nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026973(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  87nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026967(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  88nMAssay Description:Displacement of [3H]- QNB binding at the muscarinic-cholinergic binding site of rat brain S1More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026972(11-(1-Methyl-piperidin-4-ylidene)-11H-benzo[d]pyrr...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]- spiperone radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026969(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  130nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
TargetAlpha-1A adrenergic receptor(Bovine)
TBA

Curated by ChEMBL
LigandPNGBDBM50026963(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]- prazosin radioligand binding at the alpha 1-adrenergic binding site of calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026969(11-(1-Methyl-piperidin-4-ylidene)-6,11-dihydro-5H-...)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
LigandPNGBDBM50026967(11-(1-Methyl-piperidin-4-ylidene)-9-trifluoromethy...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]- apomorphine radioligand binding at the dopamine binding site of rat caudateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/13/2012
Entry Details Article
PubMed
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