Compile Data Set for Download or QSAR
Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 50035483
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50452138(CHEMBL2372196)
Affinity DataIC50: 2.40nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027512(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 4.10nMAssay Description:Inhibition of [3H]-naloxone binding to mu receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027510(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 4.80nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027508(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027508(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 5.51nMAssay Description:Inhibition of [3H]-naloxone binding to mu receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027508(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 5.51nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027506(Acetate1-(3-benzyl-2,5,8-trioxo-1,4,7triaza-cyclot...)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of [3H]-naloxone binding to mu receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027511(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 5.90nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027511(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 6.80nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027506(Acetate1-(3-benzyl-2,5,8-trioxo-1,4,7triaza-cyclot...)
Affinity DataIC50: 7.10nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027508(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 7.60nMAssay Description:Inhibitory potency against mu receptor in guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50452138(CHEMBL2372196)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027505(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 8.90nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027512(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 9.60nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027505(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 10nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027505(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 10.1nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 11nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027503(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 14nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50017233(LEVO-DROMORAN | CHEMBL592 | LEVORPHANOL)
Affinity DataIC50: 17nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50452138(CHEMBL2372196)
Affinity DataIC50: 18nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 18nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027511(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 21nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027510(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 22nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027510(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 22.4nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027509(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 23nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027511(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 23nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027503(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 24.9nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027503(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 25nMAssay Description:Inhibition of [3H]-naloxone binding to mu receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027512(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027512(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027505(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataIC50: 29nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027510(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 32nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50452138(CHEMBL2372196)
Affinity DataIC50: 48nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50027507(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 48nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 50nMAssay Description:Inhibition of [3H]-naloxone binding to mu receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027507(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 57nMAssay Description:Inhibition of [3H]-naloxone binding to mu receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027509(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 96nMAssay Description:Inhibition of [3H]-naloxone binding to mu receptor in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027506(Acetate1-(3-benzyl-2,5,8-trioxo-1,4,7triaza-cyclot...)
Affinity DataIC50: 98nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027506(Acetate1-(3-benzyl-2,5,8-trioxo-1,4,7triaza-cyclot...)
Affinity DataIC50: 98.3nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027509(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 118nMAssay Description:Inhibitory potency against Opioid receptor delta 1 in the mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027509(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 118nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to delta receptor in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027507(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 221nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50001465(2-[2-(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionyl...)
Affinity DataIC50: 246nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in the guinea pig ileum assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027503(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 253nMAssay Description:Inhibition of binding of [3H][D-Ala2,D-Leu5]enkephalin to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50017233(LEVO-DROMORAN | CHEMBL592 | LEVORPHANOL)
Affinity DataIC50: 278nMAssay Description:Inhibitory potency against Opioid receptor mu 1 in mouse vas deferens assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027507(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataIC50: 475nMAssay Description:Inhibition of [3H]naloxone binding to Opioid receptor mu 1 in rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027508(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027512(Acetate1-[1-({[1-(1-carbamoyl-3-methyl-butylcarbam...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027508(Acetate1-(6-benzyl-3-isobutyl-2,5,8,11-tetraoxo-1,...)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H][D-Ala2,D-Leu5]enkephalin binding to Opioid receptor delta 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50027506(Acetate1-(3-benzyl-2,5,8-trioxo-1,4,7triaza-cyclot...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
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