Compile Data Set for Download or QSAR
Report error Found 90 Enz. Inhib. hit(s) with all data for entry = 587
LigandPNGBDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 300nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4115(9-[(4-methanesulfonylphenyl)carbonyl]-9H-carbazole...)
Affinity DataIC50: 400nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4117(3-phenyl-1-(1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)...)
Affinity DataIC50: 400nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4100(4-[(1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)methyl]b...)
Affinity DataIC50: 400nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4109(9-(naphthalen-2-ylcarbonyl)-9H-carbazole-1,2,6,7-t...)
Affinity DataIC50: 500nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4099(9-(3-phenylpropyl)-9H-carbazole-1,2,6,7-tetrol | C...)
Affinity DataIC50: 500nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4099(9-(3-phenylpropyl)-9H-carbazole-1,2,6,7-tetrol | C...)
Affinity DataIC50: 500nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4106(9-{[4-(benzenesulfonyl)phenyl]methyl}-9H-carbazole...)
Affinity DataIC50: 600nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4108(9-[(4-phenylphenyl)carbonyl]-9H-carbazole-1,2,6,7-...)
Affinity DataIC50: 600nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4110(9-[(3-nitrophenyl)carbonyl]-9H-carbazole-1,2,6,7-t...)
Affinity DataIC50: 600nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4093(4-bromo-9H-carbazole-1,2,6,7-tetrol | Carbazole de...)
Affinity DataIC50: 600nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4078(Elagic Acid | CHEMBL6246 | 6,7,13,14-tetrahydroxy-...)
Affinity DataIC50: 600nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4113(9-[(4-tert-butylphenyl)carbonyl]-9H-carbazole-1,2,...)
Affinity DataIC50: 700nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4111(9-{[4-(trifluoromethyl)phenyl]carbonyl}-9H-carbazo...)
Affinity DataIC50: 700nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4092(9H-carbazole-1,2,6,7-tetrol | Carbazole deriv. 9b)
Affinity DataIC50: 800nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4085(2,3,8,9-tetrahydroxy-5-[(4-nitrophenyl)methyl]-5,6...)
Affinity DataIC50: 900nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4101(4-[(4-bromo-1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)...)
Affinity DataIC50: 900nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4097(9-benzoyl-9H-carbazole-1,2,6,7-tetrol | Carbazole ...)
Affinity DataIC50: 900nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4103(9-[(2,6-dichlorophenyl)methyl]-9H-carbazole-1,2,6,...)
Affinity DataIC50: 900nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4080(2,3,7,8-tetrahydroxy-5,6-dihydrophenanthridin-6-on...)
Affinity DataIC50: 900nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4109(9-(naphthalen-2-ylcarbonyl)-9H-carbazole-1,2,6,7-t...)
Affinity DataIC50: 1.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4079(2,3,8,9-tetrahydroxy-5,6-dihydrophenanthridin-6-on...)
Affinity DataIC50: 1.00E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4087(5-[(3,4-dichlorophenyl)methyl]-2,3,8,9-tetrahydrox...)
Affinity DataIC50: 1.30E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4107(9-[(4-bromophenyl)carbonyl]-9H-carbazole-1,2,6,7-t...)
Affinity DataIC50: 1.40E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4091(9H-carbazole-2,3,6,7-tetrol | Carbazole deriv. 9a)
Affinity DataIC50: 1.50E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4110(9-[(3-nitrophenyl)carbonyl]-9H-carbazole-1,2,6,7-t...)
Affinity DataIC50: 1.50E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4105(9-[(3-methylphenyl)methyl]-9H-carbazole-1,2,6,7-te...)
Affinity DataIC50: 1.70E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4112(4-bromo-9-{[4-(trifluoromethyl)phenyl]carbonyl}-9H...)
Affinity DataIC50: 2.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4089(5-{[4-(benzenesulfonyl)phenyl]methyl}-2,3,8,9-tetr...)
Affinity DataIC50: 2.00E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4095(9-benzyl-9H-carbazole-1,2,6,7-tetrol | Carbazole d...)
Affinity DataIC50: 2.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4117(3-phenyl-1-(1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)...)
Affinity DataIC50: 2.30E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4108(9-[(4-phenylphenyl)carbonyl]-9H-carbazole-1,2,6,7-...)
Affinity DataIC50: 3.20E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4104(9-[(4-bromophenyl)methyl]-9H-carbazole-1,2,6,7-tet...)
Affinity DataIC50: 3.40E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4116(4-bromo-9-[(4-methanesulfonylphenyl)carbonyl]-9H-c...)
Affinity DataIC50: 4.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4096(9-benzoyl-9H-carbazole-2,3,6,7-tetrol | Carbazole ...)
Affinity DataIC50: 4.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4081(5-ethyl-2,3,8,9-tetrahydroxy-5,6-dihydrophenanthri...)
Affinity DataIC50: 4.10E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4107(9-[(4-bromophenyl)carbonyl]-9H-carbazole-1,2,6,7-t...)
Affinity DataIC50: 4.20E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4083(5-benzyl-2,3,8,9-tetrahydroxy-5,6-dihydrophenanthr...)
Affinity DataIC50: 5.40E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4101(4-[(4-bromo-1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)...)
Affinity DataIC50: 6.60E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4094(9-benzyl-9H-carbazole-2,3,6,7-tetrol | Carbazole d...)
Affinity DataIC50: 7.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4112(4-bromo-9-{[4-(trifluoromethyl)phenyl]carbonyl}-9H...)
Affinity DataIC50: 7.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4090(5-{[4-(benzenesulfonyl)phenyl]methyl}-2,3,7,8-tetr...)
Affinity DataIC50: 7.20E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4120(9-[(2,5-dichlorobenzene)sulfonyl]-9H-carbazole-1,2...)
Affinity DataIC50: 7.70E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4098(9-(pyridin-3-ylmethyl)-9H-carbazole-2,3,6,7-tetrol...)
Affinity DataIC50: 8.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4085(2,3,8,9-tetrahydroxy-5-[(4-nitrophenyl)methyl]-5,6...)
Affinity DataIC50: 8.40E+3nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4116(4-bromo-9-[(4-methanesulfonylphenyl)carbonyl]-9H-c...)
Affinity DataIC50: 9.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4102(9-{[4-(trifluoromethyl)phenyl]methyl}-9H-carbazole...)
Affinity DataIC50: 9.00E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4111(9-{[4-(trifluoromethyl)phenyl]carbonyl}-9H-carbazo...)
Affinity DataIC50: 1.00E+4nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4082(5-ethyl-2,3,7,8-tetrahydroxy-5,6-dihydrophenanthri...)
Affinity DataIC50: 1.10E+4nMpH: 7.4 T: 2°CAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
LigandPNGBDBM4114(4-bromo-9-[(4-tert-butylphenyl)carbonyl]-9H-carbaz...)
Affinity DataIC50: 1.20E+4nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/28/2005
Entry Details Article
PubMed
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