Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50005163
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033660({[5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-pentyl]...)
Affinity DataKi:  3.10nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of zinc chlorideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033663({[6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-hexyl]-...)
Affinity DataKi:  3.70nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of zinc chlorideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033666({[2-(2-Amino-6-oxo-1,6-dihydro-purin-9-ylmethoxy)-...)
Affinity DataKi:  4.20nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of zinc chlorideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033661({[7-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-heptyl]...)
Affinity DataKi:  10nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of zinc chlorideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033666({[2-(2-Amino-6-oxo-1,6-dihydro-purin-9-ylmethoxy)-...)
Affinity DataKi:  11nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of ethylenediaminetetraacetic acid (Na2 EDTA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033664({[4-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-butyl]-...)
Affinity DataKi:  100nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of zinc chlorideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033663({[6-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-hexyl]-...)
Affinity DataKi:  390nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of ethylenediaminetetraacetic acid (Na2 EDTA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033660({[5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-pentyl]...)
Affinity DataKi:  900nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of ethylenediaminetetraacetic acid (Na2 EDTA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033665({[5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-pentyl]...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of zinc chlorideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033661({[7-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-heptyl]...)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of ethylenediaminetetraacetic acid (Na2 EDTA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033664({[4-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-butyl]-...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of ethylenediaminetetraacetic acid (Na2 EDTA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033662({Hydroxy-[5-(2-hydroxy-6-oxo-1,6-dihydro-purin-9-y...)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of zinc chlorideMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033665({[5-(2-Amino-6-oxo-1,6-dihydro-purin-9-yl)-pentyl]...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of ethylenediaminetetraacetic acid (Na2 EDTA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPurine nucleoside phosphorylase(Human)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50033662({Hydroxy-[5-(2-hydroxy-6-oxo-1,6-dihydro-purin-9-y...)
Affinity DataKi:  2.70E+5nMAssay Description:Inhibition of human erythrocyte purine nucleoside phosphorylase (PNPase) in the presence of ethylenediaminetetraacetic acid (Na2 EDTA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed