Compile Data Set for Download or QSAR
Report error Found 23 Enz. Inhib. hit(s) with all data for entry = 50005171
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033743(7-[3-(2-Cyclopropylmethyl-3-methoxy-4-thiazol-4-yl...)
Affinity DataIC50: 3.20nMAssay Description:Binding affinity towards Leukotriene B4 (LTB4) Receptor. Experiment conducted in the absence of NDGA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033744(7-{3-[3-Methoxy-2-propyl-4-(3H-[1,2,3]triazol-4-yl...)
Affinity DataIC50: 5.20nMAssay Description:Binding affinity towards Leukotriene B4 (LTB4) Receptor. Experiment conducted in the absence of NDGA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033742(3-{7-[3-(2-Cyclopropylmethyl-3-methoxy-4-thiazol-4...)
Affinity DataIC50: 12.3nMAssay Description:Binding affinity towards Leukotriene B4 (LTB4) Receptor. Experiment conducted in the absence of NDGA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033753(4-[3-(2-Cyclopropylmethyl-3-methoxy-4-thiazol-4-yl...)
Affinity DataIC50: 15.5nMAssay Description:Binding affinity towards Leukotriene B4 (LTB4) Receptor. Experiment conducted in the absence of NDGA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033747(7-[3-(2-Allyl-3-methoxy-4-thiazol-4-yl-phenoxy)-pr...)
Affinity DataIC50: 25nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033749(3-{7-[3-(3-Methoxy-2-propyl-4-thiazol-4-yl-phenoxy...)
Affinity DataIC50: 26nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033743(7-[3-(2-Cyclopropylmethyl-3-methoxy-4-thiazol-4-yl...)
Affinity DataIC50: 42nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033743(7-[3-(2-Cyclopropylmethyl-3-methoxy-4-thiazol-4-yl...)
Affinity DataIC50: 42nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50001610(CHEMBL14823 | CGS 24115 | 7-[3-(4-Acetyl-3-methoxy...)
Affinity DataIC50: 43nMAssay Description:Binding affinity towards Leukotriene B4 (LTB4) Receptor. (Experiment conducted in the absence of NDGA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033748(7-[3-(3-Methoxy-2-propyl-4-thiazol-4-yl-phenoxy)-p...)
Affinity DataIC50: 93nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033756(7-[3-(3-Methoxy-4-oxazol-4-yl-2-propyl-phenoxy)-pr...)
Affinity DataIC50: 100nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033746(SC-48928 | 7-[3-(4-Carbamoyl-3-methoxy-2-propyl-ph...)
Affinity DataIC50: 140nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033755(7-{3-[4-(2-Amino-thiazol-4-yl)-3-methoxy-2-propyl-...)
Affinity DataIC50: 320nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50001610(CHEMBL14823 | CGS 24115 | 7-[3-(4-Acetyl-3-methoxy...)
Affinity DataIC50: 320nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033750(7-{3-[4-(3H-Imidazol-4-yl)-3-methoxy-2-propyl-phen...)
Affinity DataIC50: 520nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033758(7-{3-[3-Methoxy-2-propyl-4-(1H-pyrazol-3-yl)-pheno...)
Affinity DataIC50: 610nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033745(7-{3-[4-(2-Benzylsulfanyl-1H-imidazol-4-yl)-3-meth...)
Affinity DataIC50: 750nMAssay Description:Binding affinity towards Leukotriene B4 (LTB4) Receptor. Experiment conducted in the absence of NDGA.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033757(7-[3-(4-Isoxazol-5-yl-3-methoxy-2-propyl-phenoxy)-...)
Affinity DataIC50: 770nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033752(7-{3-[4-(2-Mercapto-thiazol-4-yl)-3-methoxy-2-prop...)
Affinity DataIC50: 890nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033751(7-{3-[3-Methoxy-4-(2-methyl-oxazol-4-yl)-2-propyl-...)
Affinity DataIC50: 1.10E+3nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033754(7-{3-[3-Methoxy-4-(2-methoxy-thiazol-4-yl)-2-propy...)
Affinity DataIC50: 1.15E+3nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033759(7-{3-[3-Methoxy-4-(2-methylsulfanyl-thiazol-4-yl)-...)
Affinity DataIC50: 2.80E+3nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetLeukotriene B4 receptor 1(Human)
Searle Research and Development

Curated by ChEMBL
LigandPNGBDBM50033760(7-{3-[4-(2-Benzylsulfanyl-thiazol-4-yl)-3-methoxy-...)
Affinity DataIC50: 5.80E+3nMAssay Description:Binding affinity for Leukotriene B4 (LTB4) receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed