Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50030198
TargetVasopressin V1a receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50292418(Khusimol | CHEMBL511334)
Affinity DataIC50: 1.25E+5nMAssay Description:Displacement of [3H]AVP from vasopressin V1a receptor in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50114031(1-[5-Chloro-3-(2-chloro-phenyl)-1-(3,4-dimethoxy-b...)
Affinity DataKi:  2nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50029644(N-(3-(4-(4-(2-oxo-3,4-dihydroquinolin-1(2H)-yl)pip...)
Affinity DataKi:  350nMAssay Description:Binding affinity to vasopressin V1a receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50292418(Khusimol | CHEMBL511334)
Affinity DataKi:  4.10E+4nMAssay Description:Displacement of [3H]AVP from vasopressin V1a receptor in rat liver membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed
TargetVasopressin V1a receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50292418(Khusimol | CHEMBL511334)
Affinity DataKi:  5.30E+4nMAssay Description:Displacement of [3H]AVP from vasopressin V1a receptor in rat liver membrane by competitive displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2010
Entry Details Article
PubMed