Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50005381
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Ly...)
Affinity DataIC50: 0.580nMAssay Description:Binding affinity towards Opioid receptor kappa 1 in guinea pig brain using [3H]U-69593 as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50138774(Linear [D-Ala3]Dyn A-(1-11)NH2 | CHEMBL415795)
Affinity DataIC50: 0.760nMAssay Description:Binding affinity towards Opioid receptor kappa 1 in guinea pig brain using [3H]U-69593 as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50036266(Dyn A(H-Tyr-Gly-Ala-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Ly...)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity towards Opioid receptor kappa 1 in guinea pig brain using [3H]U-69593 as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Ly...)
Affinity DataIC50: 9.90nMAssay Description:Binding affinity towards Opioid receptor mu 1 in guinea pig brain using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50036267(Dyn A(H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Ly...)
Affinity DataIC50: 26nMAssay Description:Compound was evaluated for its receptor binding affinity at [3H]cyclo[D-pen2,p-cl-Phe4,D-Pen5](delta receptor) to opioid receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50036266(Dyn A(H-Tyr-Gly-Ala-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Ly...)
Affinity DataIC50: 210nMAssay Description:Binding affinity towards Opioid receptor mu 1 in guinea pig brain using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50138774(Linear [D-Ala3]Dyn A-(1-11)NH2 | CHEMBL415795)
Affinity DataIC50: 260nMAssay Description:Binding affinity towards Opioid receptor mu 1 in guinea pig brain using [3H]DAMGO as radioligand.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50036266(Dyn A(H-Tyr-Gly-Ala-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Ly...)
Affinity DataIC50: 730nMAssay Description:Compound was evaluated for its receptor binding affinity at [3H]cyclo[D-pen2,p-cl-Phe4,D-Pen5](delta receptor) to opioid receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50138774(Linear [D-Ala3]Dyn A-(1-11)NH2 | CHEMBL415795)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was evaluated for its receptor binding affinity at [3H]cyclo[D-pen2,p-cl-Phe4,D-Pen5](delta receptor) to opioid receptor in guinea pig brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed