Compile Data Set for Download or QSAR
Report error Found 16 Enz. Inhib. hit(s) with all data for entry = 50003382
Target5-hydroxytryptamine receptor 2A(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50469883(CHEBI:584020 | Deseril | Methysergide)
Affinity DataKi:  1.40nMAssay Description:Inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2A receptor rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409497(CHEMBL87717)
Affinity DataKi:  2.5nMAssay Description:Inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2A receptor rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409514(CHEMBL87458)
Affinity DataKi:  3.80nMAssay Description:Inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2A receptor rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]-spiperone 23390 binding to dopamine receptor D2 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409509(CHEMBL87943)
Affinity DataKi:  7.80nMAssay Description:Inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2A receptor rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409488(CHEMBL87026)
Affinity DataKi:  13nMAssay Description:Inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2A receptor rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  20nMAssay Description:Inhibition of [3H]ketanserin binding to 5-hydroxytryptamine 2A receptor rat frontal cortex membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409488(CHEMBL87026)
Affinity DataKi:  47nMAssay Description:Inhibition of [3H]-spiperone 23390 binding to dopamine receptor D2 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409514(CHEMBL87458)
Affinity DataKi:  48nMAssay Description:Inhibition of [3H]-spiperone 23390 binding to dopamine receptor D2 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409509(CHEMBL87943)
Affinity DataKi:  48nMAssay Description:Inhibition of [3H]-spiperone 23390 binding to dopamine receptor D2 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409497(CHEMBL87717)
Affinity DataKi:  71nMAssay Description:Inhibition of [3H]-spiperone 23390 binding to dopamine receptor D2 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  98nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409514(CHEMBL87458)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409488(CHEMBL87026)
Affinity DataKi:  1.29E+3nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409509(CHEMBL87943)
Affinity DataKi:  1.55E+3nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetD(1A) dopamine receptor(Rat)
University of Santiago De Compostela

Curated by ChEMBL
LigandPNGBDBM50409497(CHEMBL87717)
Affinity DataKi:  2.82E+3nMAssay Description:Inhibition of [3H]-SCH- 23390 binding to dopamine receptor D1 rat striatal membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed