Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50005456
Affinity DataKi: 0.25nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 0.570nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 76nMAssay Description:In vivo binding affinity against mu opioid receptor was measured by using labeled ligand [3H]naloxone (0.5 nM)More data for this Ligand-Target Pair
Affinity DataKi: 84nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 140nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 186nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 375nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 440nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 580nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 710nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 1.76E+3nMAssay Description:In vivo binding affinity against delta Opioid receptor was measured by using labeled ligand [3H]DADLE (1 nM) with 4 nM sufentanilMore data for this Ligand-Target Pair
Affinity DataKi: 1.87E+3nMAssay Description:In vivo binding affinity against kappa opioid receptor was measured by using labeled ligand [3H]ethylketocyclazocine (1 nM) with 500 nM DADLE and 20 ...More data for this Ligand-Target Pair
Affinity DataKi: 2.09E+3nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+5nMAssay Description:In vivo binding affinity against sigma Opioid receptor was measured by using labeled ligand [3H]-SKF- 10,047 (1 nM)More data for this Ligand-Target Pair



3D Structure (crystal)





