Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50036263
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039635(2,6-Dichloro-3-(4-methyl-piperazine-1-sulfonyl)-be...)
Affinity DataKi:  0.00700nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039646(2,6-Dichloro-3-(2-morpholin-4-yl-ethoxy)-benzoic a...)
Affinity DataKi:  0.00800nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039637(2,6-Dichloro-3-[(2-dimethylamino-ethyl)-methyl-sul...)
Affinity DataKi:  0.0100nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039631(2,6-Dichloro-benzoic acid 4-isopropyl-1,1,3-trioxo...)
Affinity DataKi:  0.0300nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039641(2,6-Dichloro-benzoic acid 4-sec-butyl-1,1,3-trioxo...)
Affinity DataKi:  0.0600nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039642(2,6-Dichloro-benzoic acid 4-ethyl-1,1,3-trioxo-1,3...)
Affinity DataKi:  0.170nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039634(2,6-Dichloro-benzoic acid 1,1,3-trioxo-4-phenyl-1,...)
Affinity DataKi:  1nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039644(2,6-Dichloro-benzoic acid 4-methyl-1,1,3-trioxo-1,...)
Affinity DataKi:  2nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039636(2,6-Dichloro-benzoic acid 1,1,3-trioxo-1,3-dihydro...)
Affinity DataKi:  2.70nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039640(2,6-Dimethyl-benzoic acid 1,1,3-trioxo-1,3-dihydro...)
Affinity DataKi:  4nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039639(2,6-Difluoro-benzoic acid 1,1,3-trioxo-1,3-dihydro...)
Affinity DataKi:  8nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039638(2,6-Dimethoxy-benzoic acid 1,1,3-trioxo-1,3-dihydr...)
Affinity DataKi:  8nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039632(2,6-Dibromo-benzoic acid 1,1,3-trioxo-1,3-dihydro-...)
Affinity DataKi:  8.5nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039633(2-Acetylamino-6-chloro-benzoic acid 1,1,3-trioxo-1...)
Affinity DataKi:  18nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039647(2,6-Dichloro-benzoic acid 4-tert-butyl-1,1,3-triox...)
Affinity DataKi:  26nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039643(Benzoic acid 1,1,3-trioxo-1,3-dihydro-1lambda*6*-b...)
Affinity DataKi:  31nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039645(2,6-Bis-trifluoromethyl-benzoic acid 1,1,3-trioxo-...)
Affinity DataKi:  37nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetNeutrophil elastase(Human)
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039648(Acetic acid 1,1,3-trioxo-1,3-dihydro-1lambda*6*-be...)
Affinity DataKi:  102nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed