Compile Data Set for Download or QSAR
Report error Found 137 Enz. Inhib. hit(s) with all data for entry = 4980
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  0.00100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82455(BIM-23027 | N-Methylcyclo[L-Ala-L-Tyr-D-Trp-L-Lys-...)
Affinity DataKi:  0.00100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84623(NC4-28B)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84626(BIM 23034)
Affinity DataKi:  0.00200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.00500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82469(EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...)
Affinity DataKi:  0.00500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82462(D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr-NH2 | BIM 2...)
Affinity DataKi:  0.00800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  0.0100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84629(BIM 23056)
Affinity DataKi:  0.0200nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82459(BIM-23058 | D-Phe-L-Phe-L-Tyr-D-Trp-L-Lys-L-Val-L-...)
Affinity DataKi:  0.0400nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.0700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82457((1R,4S,7S,10R,13S,16R)-4-[(R)-1-Hydroxyethyl]-7-(4...)
Affinity DataKi:  0.0800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  0.150nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | NSC_3086456 | MK 678)
Affinity DataKi:  0.180nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 1(Human)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50097783(SRIF-D-Trp8 | D-Trp8 SST-14 | CHEMBL438401 | SOMAT...)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataKi:  0.280nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82253(CAS_133073-82-2 | BIM 23052)
Affinity DataKi:  0.420nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50254239(somatostatin-28)
Affinity DataKi:  0.430nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84624(BIM 23068)
Affinity DataKi:  0.800nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84620(DC23-60)
Affinity DataKi:  0.930nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM85008(BIM 23066 | BIM-23066)
Affinity DataKi:  1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  1.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82469(EC5-21 | BIM-23003 | L-Cys(1)-L-Lys-L-Asn-4-Chloro...)
Affinity DataKi:  2.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84622(BIM 23057)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82455(BIM-23027 | N-Methylcyclo[L-Ala-L-Tyr-D-Trp-L-Lys-...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50059090(CHEMBL405598 | octreotide | 10-(4-Amino-butyl)-19-...)
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM85008(BIM 23066 | BIM-23066)
Affinity DataKi:  3.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84621(BIM 23042)
Affinity DataKi:  4.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50063819(CHEMBL413535 | BIM 23050 | cyclo[NMeDAla-Tyr-DTrp-...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84628(EC5-21)
Affinity DataKi:  4.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84622(BIM 23057)
Affinity DataKi:  4.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82470(3-(2-Naphtyl)-D-Ala-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-V...)
Affinity DataKi:  5.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82456(CAS_117580-24-2 | BIM 23030)
Affinity DataKi:  6.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84617(L-Alaninamide,D-phenylalanyl-L-alanyl-L-tyrosyl-D-...)
Affinity DataKi:  6.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82462(D-Nal-c[Cys-Tyr-D-Trp-Lys-Thr-Cys]-Thr-NH2 | BIM 2...)
Affinity DataKi:  7.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84638(BIM 23070)
Affinity DataKi:  7.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82466(L-362862 | c[Aha-Phe-p-C1-Phe-D-Trp-Lys-Thr-Phe] |...)
Affinity DataKi:  8.30nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 2(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKi:  8.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82458(D-Nal-Ala-Tyr-D-Trp-Lys-Val-Ala-Thr-NH2 | BIM 2304...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84619(CAS_150155-63-8 | L-Threoninamide,3-(2-naphthaleny...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM81766(CAS_3086456 | NSC_3086456 | MK 678)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82465(D-Phe-L-Cys(1)-L-Tyr-D-Trp-L-Lys-L-Abu-L-Cys(1)-L-...)
Affinity DataKi:  13.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84630(BIM 23060)
Affinity DataKi:  17.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM82454(N-Methylcyclo(D-Ala-D-Phe-D-Trp-L-Lys-D-Thr-N-meth...)
Affinity DataKi:  18.9nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
TargetSomatostatin receptor type 3(Mouse)
University of Pennsylvania

Curated by PDSP Ki Database
LigandPNGBDBM84628(EC5-21)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/2/2012
Entry Details
PubMed
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