Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 50036310
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50004477(N-(1-Carbamoyl-2-phenyl-ethyl)-3-({2-[3-(1H-indol-...)
Affinity DataIC50: 0.5nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50004474(CHEMBL316949 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{2...)
Affinity DataIC50: 0.770nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50016425(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataIC50: 0.930nMAssay Description:In vitro ability to inhibit [3H]propionyl-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50004482(CCK7 analogue | CHEMBL263742 | N-(1-Carbamoyl-2-ph...)
Affinity DataIC50: 0.990nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040523((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 3.70nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50007925(CHEMBL320868 | 3-{1-[1-aminobutyl oxycarbonylamino...)
Affinity DataIC50: 3.80nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040523((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 4.30nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50004475(CCK7 analogue | CHEMBL439591 | N-(1-Carbamoyl-2-ph...)
Affinity DataIC50: 4.70nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040520((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 5.30nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040524((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{[(S)-2-[...)
Affinity DataIC50: 14nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040522((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 16nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040518(3-{2-[2-(2-{2-[2-(tert-Butoxycarbonyl-methyl-amino...)
Affinity DataIC50: 19nMAssay Description:In vitro ability to inhibit [3H]propionyl-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040528((S)-3-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 68nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040521((S)-3-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 117nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50004490(N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2-{3-(1H-indol-3...)
Affinity DataIC50: 140nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040529((S)-3-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 170nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040520((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 427nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040525((S)-3-[(S)-2-[(S)-2-(tert-Butoxycarbonyl-methyl-am...)
Affinity DataIC50: 567nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetCholecystokinin receptor type A(Guinea pig)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040517((S)-3-{[(S)-2-[(S)-2-(tert-Butoxycarbonyl-methyl-a...)
Affinity DataIC50: 707nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type A receptor in guinea pig pancreasMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040528((S)-3-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 775nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50007925(CHEMBL320868 | 3-{1-[1-aminobutyl oxycarbonylamino...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040522((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-[(S)-2-[(...)
Affinity DataIC50: 3.72E+3nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040529((S)-3-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 4.25E+3nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040523((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 4.50E+3nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040525((S)-3-[(S)-2-[(S)-2-(tert-Butoxycarbonyl-methyl-am...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040521((S)-3-[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040523((S)-3-{[(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040517((S)-3-{[(S)-2-[(S)-2-(tert-Butoxycarbonyl-methyl-a...)
Affinity DataIC50: 1.00E+4nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50040524((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-{[(S)-2-[...)
Affinity DataIC50: 6.92E+4nMAssay Description:In vitro ability to inhibit [125I]Bolton-Hunter-CCK-8 binding to Cholecystokinin type B receptor in guinea pig cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed