Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 50005796
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataKi:  0.700nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataKi:  0.700nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041071((2-Mercaptomethyl-3-phenyl-butyrylamino)-acetic ac...)
Affinity DataIC50: 1.30nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.60nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.60nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataIC50: 2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041067(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50: 2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041069(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50: 2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041058(2-(3-Benzo[1,3]dioxol-5-yl-2-mercaptomethyl-butyry...)
Affinity DataIC50: 2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041070(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50: 2.40nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041054(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50: 2.5nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041062(3-(4-Hydroxy-phenyl)-2-[2-mercaptomethyl-3-(4-meth...)
Affinity DataIC50: 2.5nMAssay Description:In vivo inhibitory potency against Neutral Endopeptidase by measuring the displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041061(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-hexanoi...)
Affinity DataIC50: 3.10nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041053(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50: 3.5nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041059(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-4-methy...)
Affinity DataIC50: 3.5nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041062(3-(4-Hydroxy-phenyl)-2-[2-mercaptomethyl-3-(4-meth...)
Affinity DataIC50: 3.60nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041063(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-pentano...)
Affinity DataIC50: 4nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041066(3-Benzyloxy-2-(2-mercaptomethyl-3-phenyl-butyrylam...)
Affinity DataIC50: 4nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041060(2-[3-(3,4-Dimethoxy-phenyl)-2-mercaptomethyl-butyr...)
Affinity DataIC50: 4nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041063(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-pentano...)
Affinity DataIC50: 4nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041054(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50: 4.30nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041057(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50: 4.5nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041053(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50: 5nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041057(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50: 5.20nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407298(CHEMBL2051772)
Affinity DataKi:  5.30nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041052(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-butyric...)
Affinity DataIC50: 5.40nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041064(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50: 5.90nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041052(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-butyric...)
Affinity DataIC50: 6.30nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041064(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50: 6.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041061(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-hexanoi...)
Affinity DataIC50: 7nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041068(3-(4-Hydroxy-phenyl)-2-[3-(4-hydroxy-phenyl)-2-mer...)
Affinity DataIC50: 7.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041068(3-(4-Hydroxy-phenyl)-2-[3-(4-hydroxy-phenyl)-2-mer...)
Affinity DataIC50: 9nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041058(2-(3-Benzo[1,3]dioxol-5-yl-2-mercaptomethyl-butyry...)
Affinity DataIC50: 9.5nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407298(CHEMBL2051772)
Affinity DataKi:  10nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041067(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50: 10nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041050(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-o-tolyl...)
Affinity DataIC50: 11nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041055(2-[3-(4-Amino-phenyl)-2-mercaptomethyl-butyrylamin...)
Affinity DataIC50: 12nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041051(2-[3-(4-Hydroxy-3-methoxy-phenyl)-2-mercaptomethyl...)
Affinity DataIC50: 14nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041065(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-3-methy...)
Affinity DataIC50: 15nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041060(2-[3-(3,4-Dimethoxy-phenyl)-2-mercaptomethyl-butyr...)
Affinity DataIC50: 16nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041055(2-[3-(4-Amino-phenyl)-2-mercaptomethyl-butyrylamin...)
Affinity DataIC50: 16nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataKi:  16nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041059(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-4-methy...)
Affinity DataIC50: 19nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataIC50: 20nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041069(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50: 25nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041071((2-Mercaptomethyl-3-phenyl-butyrylamino)-acetic ac...)
Affinity DataIC50: 32nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAngiotensin-converting enzyme(Mouse)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041066(3-Benzyloxy-2-(2-mercaptomethyl-3-phenyl-butyrylam...)
Affinity DataIC50: 43nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeprilysin(Human)
University of Paris

Curated by ChEMBL
LigandPNGBDBM50041051(2-[3-(4-Hydroxy-3-methoxy-phenyl)-2-mercaptomethyl...)
Affinity DataIC50: 65nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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