Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50036233
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50: 18nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50: 42nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50: 66nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50: 85nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 570nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 620nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50: 760nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50: 760nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudinal muscle-myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 7.30E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudinal muscle-myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50: 1.10E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50: 1.20E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50: 2.25E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudinal muscle-myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50: 3.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50: 3.30E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Mouse)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50: 3.30E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudinal muscle-myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(CHEMBL294616 | 13-[2-Amino-3-(4-hydroxy-phenyl)-pr...)
Affinity DataIC50: 3.50E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50: 3.90E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudinal muscle-myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50: 5.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Rat)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50: 5.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetMu-type opioid receptor(Guinea pig)
University of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudinal muscle-myenteric plexusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed