Report error Found 61 Enz. Inhib. hit(s) with all data for entry = 50005880
Affinity DataIC50: 6nMAssay Description:Binding effinity for sigma receptor using 2 nM of [3H]DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding effinity for sigma receptor using 2 nM of [3H]-DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Binding effinity for sigma receptor using 2 nM of [3H]DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Binding effinity for sigma receptor using 2 nM of [3H]DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 430nMAssay Description:Binding effinity for sigma receptor using 2 nM of [3H]DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 520nMAssay Description:Binding affinity for sigma receptor using 2 nM of [3H]DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Binding effinity for sigma receptor using 2 nM of [3H]DTG as radioligand, in membranes from brain minus cerebellumMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding towards Dopamine receptor D2 using [3H]spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Evaluated for binding towards dopamine D2-receptor using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]U-86170More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 6.40nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]U-86170More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding towards Dopamine receptor D2 expressed in CHO-K1 cells using [3H]U-86170More data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Evaluated for binding towards dopamine D2-receptor using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding towards Dopamine receptor D2 using [3H]spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Evaluated for binding towards dopamine D2-receptor using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Evaluated for binding towards dopamine D2-receptor using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 158nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 217nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 249nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]N-0437 as radioligand from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Binding towards Dopamine receptor D2 using [3H]spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Binding towards Dopamine receptor D2 using [3H]spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding towards Dopamine receptor D2 using [3H]spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Binding towards Dopamine receptor D2 using [3H]spiperone from rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 776nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 776nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 889nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 889nMAssay Description:Evaluated for binding towards Dopamine receptor D2 using [3H]-spiperone as radioligand, in cloned mammalian receptors expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >933nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: >933nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: >933nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: >933nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding towards dopamine receptor D4 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
Affinity DataKi: >1.43E+3nMAssay Description:Binding towards Dopamine receptor D3 expressed in CHO-K1 cells using [3H]spiperone More data for this Ligand-Target Pair
