Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50006064
Target5-hydroxytryptamine receptor 1A(Mouse)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044237(R-(+)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Mouse)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044238(S-(-)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035320(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  0.200nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035320(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  1.30nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044237(R-(+)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  1.40nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044238(S-(-)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  2nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50016777(7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-ol...)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT (agonist) as radioligand (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035330(R-(+)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  7nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50011247(S-(-)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthale...)
Affinity DataKi:  8.40nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  8.70nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]8-OH-DPAT (agonist) as radioligand (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035329((+/-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  12nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035307(S-(-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  14nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044237(R-(+)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity against dopamine receptor D2 using [3H]raclopride as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044236(R-(+)-Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  25nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035320(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  40nMAssay Description:In vitro binding affinity against dopamine receptor D2 using [3H]-Raclopride as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50017520((+/-)-Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  66nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035330(R-(+)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035320(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  120nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035307(S-(-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  146nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50035329((+/-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  156nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044236(R-(+)-Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  170nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044235(S-(-)-Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  190nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50017520((+/-)-Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50037271(Dipropyl-(5,6,7,8-tetrahydro-1H-benzo[f]indol-7-yl...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044237(R-(+)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  382nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044238(S-(-)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  423nMAssay Description:In vitro binding affinity against dopamine receptor D2 using [3H]raclopride as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50037271(Dipropyl-(5,6,7,8-tetrahydro-1H-benzo[f]indol-7-yl...)
Affinity DataKi:  570nMAssay Description:In vitro binding affinity against 5-hydroxytryptamine 1A receptor using [3H]-8-OH-DPAT as radioligand in CHO cells (sc)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50016777(7-Dipropylamino-5,6,7,8-tetrahydro-naphthalen-1-ol...)
Affinity DataKi:  826nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataKi:  1.36E+3nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044235(S-(-)-Dimethyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  1.58E+3nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50044238(S-(-)-1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  3.59E+3nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of GöTeborg

Curated by ChEMBL
LigandPNGBDBM50011247(S-(-)-7-Dipropylamino-5,6,7,8-tetrahydro-naphthale...)
Affinity DataKi:  5.07E+3nMAssay Description:Displacement of [3H]spiperone from dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed