Report error Found 392 Enz. Inhib. hit(s) with all data for entry = 50006190
Affinity DataKi: 2.30nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9.70nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 96nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 100nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 135nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 156nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 202nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 211nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 216nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 216nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 304nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 323nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 328nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 338nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 350nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 476nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 678nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataKi: 800nMAssay Description:Binding affinity against mitochondrial DBI complex (peripheral benzodiazepine receptor) using primary cultures of glial cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]ketanserin from serotonin receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]L-365260 from cholecystokinin receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]ketanserin from serotonin receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]ketanserin from serotonin receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]ketanserin from serotonin receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [125I]pindolol from beta-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Mayo Foundation
Curated by ChEMBL
Mayo Foundation
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]clonidine from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor/Alpha-1B adrenergic receptor/Alpha-1D adrenergic receptor/Alpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(Rat)
Mayo Foundation
Curated by ChEMBL
Mayo Foundation
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [3H]clonidine from alpha-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]ketanserin from serotonin receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]L-365260 from cholecystokinin receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [125I]pindolol from beta-adrenergic receptor in rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibitory activity by measuring its ability to displace [3H]ketanserin from serotonin receptor in rat brainMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor/Kappa-type opioid receptor/Mu-type opioid receptor/Sigma non-opioid intracellular receptor 1(Rat)
Mayo Foundation
Curated by ChEMBL
Mayo Foundation
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of [3H]naxolone binding to opiate receptors in rat brainMore data for this Ligand-Target Pair







































